SCHEMBL2669953

SCHEMBL2669953

CCCCCC(C)C(Nc1ccc(C(=O)N(C)CCC(=O)O)cc1)c1oc2ccc(-c3ccc(OC)nc3)cc2c1C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BTK Q06187 8/20 0.41
TAAR1 Q96RJ0 1/20 0.37
MAPT P10636 1/20 0.37
RCE1 Q9Y256 1/20 0.36
PIK3CA P42336 6/20 0.35
HDAC1 Q13547 6/20 0.35
GCG P01275 1/20 0.35
GCGR P47871 1/20 0.34
OXTR P30559 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CB P42338 1/20 0.33
MTOR P42345 1/20 0.33
PIK3CG P48736 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL719610 0.92 BTK (0.44) BTKTAAR1MAPTRCE1PIK3CA
SCHEMBL2669960 0.88 GCG (0.40) GCGGCGR
SCHEMBL720184 0.86 BTK (0.42) BTKTAAR1MAPTRCE1PIK3CA
SCHEMBL2669834 0.86 GCG (0.41) BTKGCGGCGR
SCHEMBL2669769 0.85 NAMPT (0.36) HDAC1GCGPIK3CBHDAC6
SCHEMBL2669939 0.83 NPC1 (0.39)
SCHEMBL9070790 0.83 NAMPT (0.34) MAPTGCG
SCHEMBL13069831 0.83 NPC1 (0.33)
SCHEMBL9070778 0.82 PTGS2 (0.42) GCGHDAC6
SCHEMBL2669958 0.82 CASP3 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110520-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2009-09-11 WO disclosed