SCHEMBL2676256

SCHEMBL2676256

c1ccc2c(c1)CCNC2c1cccc2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRCP P42785 8/20 0.59
GAA P10253 1/20 0.57
RECQL P46063 1/20 0.53
GID4 Q8IVV7 1/20 0.49
MAPT P10636 2/20 0.46
SLC22A1 O15245 1/20 0.45
TSHR P16473 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KDM1A O60341 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20722382 0.91 PRCP (0.53) PRCPGAARECQLGID4MAPT
SCHEMBL4399590 0.86 GAA (0.54) PRCPGAARECQLGID4MAPT
SCHEMBL6986104 0.79 PRCP (0.52) PRCPGAARECQLGID4MAPT
SCHEMBL26116236 0.79 RECQL (0.52) PRCPGAARECQLGID4MAPT
SCHEMBL4120535 0.79 PRCP (0.50) PRCPGAARECQLGID4MAPT
SCHEMBL23274866 0.76 PRCP (0.61) PRCPGAARECQLGID4MAPT
SCHEMBL29924130 0.76 PRCP (0.61) PRCPGAARECQLGID4MAPT
SCHEMBL3068128 0.76 PRCP (0.54) PRCPGAARECQLGID4HTR2A
SCHEMBL6185636 0.75 PRCP (0.60) PRCPGAASLC22A1SMN1; SMN2
SCHEMBL6229660 0.75 PRCP (0.65) PRCPGAARECQLGID4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4659812-A1 DETECTION METHODS AND COMBINATION THERAPIES OF CELLS WITH EXTRACELLULAR RAS EXPRESSION Bumm, Thomas (DE) 2025-12-10 EP disclosed
US-20230132973-A1 DIHYDRO-SPIRO[INDOLINE-3:1'-iSOQUINOLIN]-2-ONES AS ANTIMALARIAL AGENTS THE UNIV OF BUEA (CM) 2023-05-04 US disclosed
WO-2021186348-A1 DIHYDRO-SPIRO[INDOLINE-3:1'-ISOQUINOLIN]-2-ONES AS ANTIMALARIAL AGENTS THE UNIVERSITY OF BUEA (CM) 2021-09-23 WO disclosed
EP-2074100-B1 BIOFILM-INHIBITING EFFECT AND ANTI-INFECTIVE ACTIVITY OF N,C-LINKED ARYLISOQUINOLINES AND THE USE THEREOF UNIV WUERZBURG J MAXIMILIANS (DE) 2013-08-28 EP disclosed
US-8173673-B2 Biofilm-inhibiting effect and anti-infective activity of N,C-linked aryl isoquinolines and the use thereof JULIUS-MAXIMILIANS-UNIVERSITAET WUERZBURG (DE) 2012-05-08 US disclosed
US-20100286198-A1 Biofilm-Inhibiting Effect and Anti-Infective Activity of N,C- Linked Arylisoquinolines and the Use Thereof JULIUS-MAXIMILIANS-UNIVERSITAET WUERZBURG (DE) 2010-11-11 US disclosed
EP-2074100-A1 BIOFILM-INHIBITING EFFECT AND ANTI-INFECTIVE ACTIVITY OF N,C-LINKED ARYLISOQUINOLINES AND THE USE THEREOF Julius-Maximilians-Universität Würzburg (DE) 2009-07-01 EP disclosed
WO-2008037482-A1 BIOFILM-INHIBITING EFFECT AND ANTI-INFECTIVE ACTIVITY OF N,C-LINKED ARYLISOQUINOLINES AND THE USE THEREOF JULIUS-MAXIMILIANS-UNIVERSITÄT WÜRZBURG (DE) 2008-04-03 WO disclosed
EP-1045837-B1 MONOMERIC AND DIMERIC ARYLISOQUINOLINE ALKALOIDS AND DERIVATIVES THEREOF US GOV HEALTH & HUMAN SERV (US) 2007-03-14 EP disclosed
US-6331630-B1 Dimeric arylisoquinoline alkaloids and derivatives thereof THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2001-12-18 US disclosed
US-6140339-A Monomeric and dimeric arylisoquinoline alkaloids and derivatives thereof THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-10-31 US disclosed
EP-1045837-A1 MONOMERIC AND DIMERIC ARYLISOQUINOLINE ALKALOIDS AND DERIVATIVES THEREOF THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-10-25 EP disclosed
WO-1999033811-A1 MONOMERIC AND DIMERIC ARYLISOQUINOLINE ALKALOIDS AND DERIVATIVES THEREOF THE GOVERNMENT OF THE UNITED STATES OF AMERICA, R EPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1999-07-08 WO disclosed
EP-0745066-A1 ANTIMALARIAL KORUPENSAMINES AND PHARMACEUTICAL COMPOSITIONS AND MEDICAL USES THEREOF THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1996-12-04 EP disclosed
WO-1995021826-A1 ANTIMALARIAL KORUPENSAMINES AND PHARMACEUTICAL COMPOSITIONS AND MEDICAL USES THEREOF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-08-17 WO disclosed
US-5409938-A A plant extracts having a naphthyl-tetrahydroisoquinolines group; a new drug treating malarial, parasiticides THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-04-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100286198-A1 Biofilm-Inhibiting Effect and Anti-Infective Activity of N,C- Linked Arylisoquinolines and the Use Thereof PGLS, NACA, PFAS PRCP 1603/4885GAA 668/4885RECQL 478/4885
US-20230132973-A1 DIHYDRO-SPIRO[INDOLINE-3:1'-iSOQUINOLIN]-2-ONES AS ANTIMALARIAL AGENTS QDPR, NQO1, IDO2 PRCP 2729/4885GAA 3964/4885RECQL 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.