SCHEMBL2679428

SCHEMBL2679428

CNc1nccc(-c2cc(NCC(=O)NCCOC(C)C)c3cc(OC)ccc3c2)n1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 12/20 0.38
MTNR1B P49286 12/20 0.38
HDAC3 O15379 1/20 0.35
NCOR1 O75376 1/20 0.35
HDAC2 Q92769 1/20 0.35
GSK3B P49841 1/20 0.34
THRB P10828 1/20 0.34
DYRK1A Q13627 3/20 0.34
CLK4 Q9HAZ1 3/20 0.34
DYRK1B Q9Y463 3/20 0.34
CLK1 P49759 2/20 0.34
CLK2 P49760 2/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2678527 0.92 MTNR1A (0.39) MTNR1AMTNR1BHDAC3NCOR1HDAC2
SCHEMBL2678412 0.90 MTNR1A (0.40) MTNR1AMTNR1BHDAC3NCOR1HDAC2
SCHEMBL2678111 0.90 MTNR1A (0.40) MTNR1AMTNR1BHDAC3NCOR1HDAC2
SCHEMBL6128583 0.87 HDAC3 (0.35) MTNR1AMTNR1BHDAC3NCOR1HDAC2
SCHEMBL2678816 0.85 JAK2 (0.39) MTNR1AMTNR1B
SCHEMBL2679375 0.84 HDAC3 (0.41) HDAC3NCOR1HDAC2GSK3BDYRK1A
SCHEMBL2679402 0.83 MAPK9 (0.37) MTNR1AMTNR1BHDAC3NCOR1HDAC2
SCHEMBL2679029 0.83 SYK (0.48) MTNR1AMTNR1B
SCHEMBL2678213 0.83 ACHE (0.42)
SCHEMBL2678820 0.82 MEN1 (0.42) HDAC3NCOR1HDAC2GSK3BPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8173808-B2 Substituted naphthalenyl-pyrimidine compounds ARQULE, INC. (US) 2012-05-08 US claimed