SCHEMBL26802

SCHEMBL26802

O=CN(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
TSHR P16473 2/20 0.48
CA2 P00918 1/20 0.45
AOC3 Q16853 1/20 0.44
ADH1B P00325 1/20 0.43
ADH1C P00326 1/20 0.43
ADH1A P07327 1/20 0.43
ADH7 P40394 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
G6PC1 P35575 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
LMNA P02545 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5542200 0.88 KCNA5 (0.50) ALDH1A1RAB9ATDP1KDM4EMEN1
SCHEMBL5548405 0.88 G6PC1 (0.49) G6PC1TDP1KDM4EMEN1MAPT
Malonic Acid SCHEMBL16431221 0.88 NPC1 (0.47) ALDH1A1TSHRNPC1RAB9ACA12
SCHEMBL5540778 0.88 L3MBTL1 (0.45) ALDH1A1TSHRRAB9ALMNAMEN1
SCHEMBL7087904 0.87 TSHR (0.41) ALDH1A1TSHRCA2AOC3NPC1
SCHEMBL968495 0.87 LMNA (0.48) ALDH1A1TSHRAOC3NPC1RAB9A
SCHEMBL28517819 0.86 MEN1 (0.46) ALDH1A1TSHRCA2NPC1RAB9A
SCHEMBL5522932 0.85 TAAR1 (0.47) ALDH1A1TSHRAOC3NPC1RAB9A
SCHEMBL5522934 0.85 TAAR1 (0.47) ALDH1A1TSHRAOC3NPC1RAB9A
SCHEMBL9827242 0.83 HTT (0.42) ALDH1A1TSHRNPC1RAB9ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 588 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929668-B (Meth) acrylate compound having isocyanate group and method for producing same 株式会社力森诺科 2024-08-20 CN claimed
US-20230056109-A1 (METH)ACRYLIC ACID ESTER COMPOUND HAVING ISOCYANATE GROUP AND METHOD FOR PRODUCING SAME SHOWA DENKO K.K. (JP) 2023-02-23 US claimed
EP-4089070-A1 (METH)ACRYLIC ACID ESTER COMPOUND HAVING ISOCYANATE GROUP, AND METHOD FOR PRODUCING SAME Showa Denko K.K. (JP) 2022-11-16 EP claimed
CN-114929668-A (meth) acrylate compound having isocyanate group and method for producing same 昭和电工株式会社 2022-08-19 CN claimed
CN-114585611-A Triazinane derivative and process for producing the same 弗雷克斯系统美国公司 2022-06-03 CN claimed
WO-2021141002-A1 (METH)ACRYLIC ACID ESTER COMPOUND HAVING ISOCYANATE GROUP, AND METHOD FOR PRODUCING SAME 昭和電工株式会社 2021-07-15 WO claimed
EP-3027591-B1 NOVEL DERIVATIVES OF A 3,4-DIHYDROISOQUINOLINE-3-CARBOXYLIC ACID HAVING ANTI-CANCER PROPERTIES, A METHOD FOR THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAID DERIVATIVES, AND THEIR USE NARODOWY INSTYTUT ZDROWIA PUBLICZNEGO PANSTWOWY ZAKL HIGIENY (PL) 2018-07-18 EP claimed
EP-2867202-B1 METHOD FOR PRODUCING STEREOSELECTIVE EPOXYKETONE COMPOUND NISSAN CHEMICAL IND LTD (JP) 2017-08-09 EP claimed
US-20170036993-A1 METAL-ORGANIC FRAMEWORK FOR FLUID STREAM FILTRATION APPLICATIONS EASTMAN CHEMICAL COMPANY (US) 2017-02-09 US claimed
EP-2423212-B1 PROCESS FOR PRODUCTION OF 2-AZAADAMANTANE COMPOUND FROM BICYCLOCARBAMATE COMPOUND NISSAN CHEMICAL IND LTD (JP) 2016-06-01 EP claimed
WO-1997048695-A1 NEW PYRIDYL ALKANE ACID AMIDES AS CYTOSTATICS AND IMMUNOSUPPRESSIVES KLINGE PHARMA GMBH (DE) 1997-12-24 WO claimed
WO-1997048397-A1 USE OF PYRIDYL ALKANE, PYRIDYL ALKENE AND/OR PYRIDYL ALKINE ACID AMIDES IN THE TREATMENT OF TUMORS OR FOR IMMUNOSUPPRESSION KLINGE PHARMA GMBH (DE) 1997-12-24 WO claimed
WO-1997048696-A1 PYRIDYL ALKENE- AND PYRIDYL ALKINE- ACID AMIDES AS CYTOSTATICS AND IMMUNOSUPPRESSIVES KLINGE PHARMA GMBH (DE) 1997-12-24 WO claimed
CN-1113237-A N- (2-amino-4, 6-dichloropyrimidin-5-yl) formamide and preparation method thereof LONZA AG (CH) 1995-12-13 CN claimed
EP-0684236-A2 N-(2-Amino-4,6-dichloropyrimidin-5-yl)formamide and process for its production LONZA AG (CH) 1995-11-29 EP claimed
EP-0230224-B1 PROCESS FOR THE PREPARATION OF ALCOXYCARBONYL ISOCYANATES BAYER AG (DE) 1991-07-17 EP claimed
US-4777283-A Process for the preparation of alkoxycarbonyl isocyanates BAYER AKTIENGESELLSCHAFT (DE) 1988-10-11 US claimed
EP-0115954-B1 BICYCLOOCTANE DERIVATIVES AND THEIR PRODUCTION AND USE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1987-08-19 EP claimed
EP-0230224-A2 Process for the preparation of alcoxycarbonyl isocyanates BAYER AG (DE) 1987-07-29 EP claimed
EP-0115954-A2 Bicyclooctane derivatives and their production and use SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1984-08-15 EP claimed