SCHEMBL268458

SCHEMBL268458

COC(=O)c1c(NC(=O)c2ccc(OC)c(OC)c2)sc(O)c1C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 5/20 0.65
MAPT P10636 5/20 0.54
RXFP1 Q9HBX9 3/20 0.54
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
RECQL P46063 1/20 0.54
TP53 P04637 1/20 0.53
KDM4E B2RXH2 5/20 0.53
ALDH1A1 P00352 7/20 0.52
HPGD P15428 3/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
POLB P06746 1/20 0.52
PKM P14618 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HTT P42858 2/20 0.50
GAA P10253 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
LMNA P02545 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7002672 0.79 FLT3 (1.00) FLT3MAPTKMT2AMEN1RECQL
SCHEMBL26308284 0.78 MAPT (0.64) FLT3MAPTKMT2AMEN1RECQL
SCHEMBL268017 0.78 KDM4E (0.63) FLT3MAPTRXFP1KMT2AMEN1
SCHEMBL26307731 0.78 THRB (0.68) FLT3MAPTRXFP1KMT2AMEN1
SCHEMBL267190 0.73 FLT3 (0.81) FLT3MAPTRXFP1KMT2AMEN1
SCHEMBL5788877 0.72 MAPT (0.60) FLT3MAPTKMT2AMEN1RECQL
SCHEMBL25195878 0.72 KMT2A (0.57) FLT3MAPTRXFP1KMT2AMEN1
SCHEMBL30500223 0.72 KMT2A (0.57) FLT3MAPTRXFP1KMT2AMEN1
SCHEMBL266561 0.72 KMT2A (0.58) FLT3MAPTRXFP1KMT2AMEN1
SCHEMBL267990 0.72 KDM4E (0.58) FLT3MAPTRXFP1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120115851-A1 COMPOUND INHIBITING IN VIVO PHOSPHORUS TRANSPORT AND MEDICINE CONTAINING THE SAME KYOWA HAKKO KIRIN CO., LTD. (JP) 2012-05-10 US disclosed
US-8134015-B2 Compound inhibiting in vivo phosphorous transport and medicine containing the same KYOWA HAKKO KIRIN CO., LTD. (JP) 2012-03-13 US disclosed
US-20060217426-A1 Compound inhibiting in vivo phosphorous transport and medicine containing the same KIRIN BEER KABUSHIKI KAISHA (JP) 2006-09-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060217426-A1 Compound inhibiting in vivo phosphorous transport and medicine containing the same SLC10A6, SLC7A1, SLC10A1 FLT3 1555/4885MAPT 4195/4885RXFP1 253/4885
US-20120115851-A1 COMPOUND INHIBITING IN VIVO PHOSPHORUS TRANSPORT AND MEDICINE CONTAINING THE SAME SLC34A1, SLC34A2, SLC20A2 FLT3 2535/4885MAPT 4648/4885RXFP1 295/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.