SCHEMBL26865331

SCHEMBL26865331

COc1nccc2c(Nc3ccc(S(=N)(=O)NC[C@@H](C)O)cc3)ccnc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.36
GAK O14976 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
CDK1 P06493 7/20 0.33
CDK2 P24941 7/20 0.33
KDR P35968 7/20 0.33
CCNB1 P14635 1/20 0.33
CCNE1 P24864 1/20 0.33
HTT P42858 1/20 0.33
RIPK1 Q13546 2/20 0.32
PDGFRA P16234 1/20 0.32
RIPK2 O43353 1/20 0.32
RIPK3 Q9Y572 1/20 0.32
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26656440 1.00 BRAF (0.36) BRAFGAKPTGS1PTGS2CDK1
SCHEMBL30666120 1.00 BRAF (0.36) BRAFGAKPTGS1PTGS2CDK1
SCHEMBL26864188 1.00 BRAF (0.36) BRAFGAKPTGS1PTGS2CDK1
SCHEMBL26864929 0.90 ALDH1A1 (0.35) BRAFGAKPTGS1PTGS2CDK1
SCHEMBL26863549 0.90 GAK (0.33) GAKPTGS1PTGS2CDK1CDK2
SCHEMBL26863383 0.89 PTGS1 (0.34) GAKPTGS1PTGS2CDK1CDK2
SCHEMBL26863546 0.88 BRAF (0.35) BRAFALDH1A1MAPTMTNR1A
SCHEMBL25465686 0.87 HTR1A (0.47) GAKHTTPDGFRAALDH1A1GAA
SCHEMBL26863377 0.83 GAK (0.39) GAKPTGS1PTGS2KDRHTT
SCHEMBL26862953 0.83 IKBKB (0.38) BRAFGAKPTGS1PTGS2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023225001-A1 NAPHTHYRIDINE BASED ENPP1 MODULATORS AND USES THEREOF Vir Biotechnology, Inc. (US) 2023-11-23 WO disclosed