SCHEMBL26953243

SCHEMBL26953243

NCc1ccc(-c2ccnc3[nH]cc(-c4cccnc4)c23)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.55
ROCK2 O75116 4/20 0.52
ROCK1 Q13464 4/20 0.52
CDC42BPB Q9Y5S2 3/20 0.52
CDC42BPA Q5VT25 2/20 0.51
SGK1 O00141 1/20 0.50
LRRK2 Q5S007 4/20 0.49
MAPK1 P28482 1/20 0.46
LOXL2 Q9Y4K0 1/20 0.46
NUDT1 P36639 1/20 0.46
DYRK1A Q13627 3/20 0.46
NTRK1 P04629 1/20 0.46
PIK3CA P42336 1/20 0.46
VHL P40337 1/20 0.45
MKNK2 Q9HBH9 2/20 0.44
MKNK1 Q9BUB5 1/20 0.44
CCNK O75909 1/20 0.44
CDK12 Q9NYV4 1/20 0.44
JAK3 P52333 1/20 0.44
DYRK1B Q9Y463 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31734861 1.00 CYP2A6 (0.55) CYP2A6ROCK2ROCK1CDC42BPBCDC42BPA
SCHEMBL26953278 0.90 SGK1 (0.57) CYP2A6ROCK2ROCK1CDC42BPASGK1
SCHEMBL31735012 0.90 SGK1 (0.57) CYP2A6ROCK2ROCK1CDC42BPASGK1
SCHEMBL26953219 0.83 LRRK2 (0.45) ROCK2ROCK1CDC42BPASGK1LRRK2
SCHEMBL31735137 0.83 LRRK2 (0.45) ROCK2ROCK1CDC42BPASGK1LRRK2
SCHEMBL31734890 0.83 LRRK2 (0.59) SGK1LRRK2NUDT1STK3
SCHEMBL31734958 0.83 CDK2 (0.53) ROCK2SGK1LRRK2JAK3CDC7
SCHEMBL31735005 0.83 LRRK2 (0.59) SGK1LRRK2JAK3CDK2CDK9
SCHEMBL26953170 0.83 LRRK2 (0.59) SGK1LRRK2JAK3CDK2CDK9
SCHEMBL26953245 0.83 CDK2 (0.53) ROCK2SGK1LRRK2JAK3CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023239727-A1 LATS INHIBITORS AND USES THEREOF THE USA, AS REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2023-12-14 WO disclosed