SCHEMBL26964483

SCHEMBL26964483

CCOC(=O)c1nn(COCC[Si](C)(C)C)cc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
MAPT P10636 2/20 0.42
LMNA P02545 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
MITF O75030 1/20 0.40
HTT P42858 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KCNMA1 Q12791 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22773500 0.89 ALDH1A1 (0.43) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL4016651 0.85 ALDH1A1 (0.43) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL30079506 0.85 ALDH1A1 (0.43) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL24537117 0.83 ALDH1A1 (0.40) ALDH1A1MAPTLMNASMN1; SMN2ADORA3
SCHEMBL7515726 0.82 ALDH1A1 (0.60) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL31074656 0.82 L3MBTL1 (0.45) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL18131250 0.81 MAPT (0.39) ALDH1A1MAPTLMNAPOLBPTGS1
SCHEMBL27139104 0.81 ALDH1A1 (0.35) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL15726277 0.81 NPC1 (0.37) ALDH1A1MAPTLMNASMN1; SMN2ADORA3
SCHEMBL26964472 0.81 ADORA3 (0.41) ALDH1A1MAPTLMNASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023242228-A1 4-SUBSTITUTED (1H-BENZO[D]IMIDAZOL-2-YL)-1H-PYRAZOLES AS BUB1 INHIBITORS USEFUL FOR TREATING CANCERS UNIVERSITEIT LEIDEN (NL) 2023-12-21 WO disclosed
EP-4293019-A1 4-SUBSTITUTED (1H-BENZO[D]IMIDAZOL-2-YL)-1H-PYRAZOLES AS BUB1 INHIBITORS USEFUL FOR TREATING CANCERS Netherlands Translational Research Center Holding B.V. (NL) 2023-12-20 EP disclosed