Dihydromorphine

Dihydromorphine

SCHEMBL2696539

CN1CC[C@]23c4c5ccc(O)c4OC2C(O)CC[C@H]3[C@H]1C5

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 7/20 0.71
OPRK1 P41145 6/20 0.71
OPRM1 P35372 6/20 0.71
MRGPRX2 Q96LB1 2/20 0.64
SLC22A1 O15245 1/20 0.64
ADRA2A P08913 1/20 0.64
ARRB1 P49407 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dihydromorphine SCHEMBL12402795 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL29394226 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL19107002 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL13348852 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL26346 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL19645038 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL13380388 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL19615483 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL17025853 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL15449768 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140271835-A1 ABUSE RESISTANT CAPSULE ARES CAPITAL CORPORATION, AS COLLATERAL AGENT 2014-09-18 US claimed
US-20100221322-A1 Abuse-Resistant Pharmaceutical Dosage Form GRUENENTHAL GMBH (DE) 2010-09-02 US claimed
US-20050186139-A1 Abuse-proofed dosage form GRUENENTHAL GMBH (DE) 2005-08-25 US claimed
US-20230330044-A1 METHODS AND COMPOSITIONS FOR INTERFERING WITH EXTRACTION OR CONVERSION OF A DRUG SUSCEPTIBLE TO ABUSE ACURA PHARMACEUTICALS INC (US) 2023-10-19 US disclosed
US-11224576-B2 Process for the production of an abuse-proofed dosage form Grünenthal GmbH (DE) 2022-01-18 US disclosed
EP-3824878-A1 ABUSE RESISTANT CAPSULE R.P. Scherer Technologies, LLC (US) 2021-05-26 EP disclosed
US-20200215053-A1 ABUSE-PROOFED DOSAGE FORM Grünenthal GmbH (DE) 2020-07-09 US disclosed
US-10653776-B2 Compositions and methods for reducing overdose INTELLIPHARMACEUTICS CORP. (CA) 2020-05-19 US disclosed
US-10610497-B2 Methods and compositions for interfering with extraction or conversion of a drug susceptible to abuse ACURA PHARMACEUTICALS, INC. (US) 2020-04-07 US disclosed
US-20190321358-A1 ABUSE-PROOFED DOSAGE FORM Grünenthal GmbH (DE) 2019-10-24 US disclosed
US-10420729-B2 Abuse resistant capsule R.P. SCHERER TECHNOLOGIES, LLC (US) 2019-09-24 US disclosed
US-20090004267-A1 Dosage Form with Impeded Abuse GRUENENTHAL GMBH (DE) 2009-01-01 US disclosed
US-20090005408-A1 PROCESS FOR THE PRODUCTION OF AN ABUSE-PROOFED DOSAGE FORM GRUNENTHAL GMBH (DE) 2009-01-01 US disclosed
US-20080311049-A1 Thermoforming by extrusion without discoloration; controlled release GRUNENTHAL GMBH (DE) 2008-12-18 US disclosed
US-20080311197-A1 PROCESS FOR THE PRODUCTION OF AN ABUSE-PROOFED DOSAGE FORM GRUNENTHAL GMBH (DE) 2008-12-18 US disclosed
US-20080152595-A1 Methods and compositions for deterring abuse of orally administered pharmaceutical products ACURA PHARMACEUTICALS, INC. 2008-06-26 US disclosed
US-20070003616-A1 Process for the production of an abuse-proofed dosage form ENDO PHARMACEUTICALS, INC. 2007-01-04 US disclosed
US-20050249792-A1 Active ingredient release system comprising a plaster containing an active ingredient and at least one active ingredient release regulator GRUENENTHAL GMBH (DE) 2005-11-10 US disclosed
US-20050186139-A1 Abuse-proofed dosage form GRUENENTHAL GMBH (DE) 2005-08-25 US disclosed
US-20050031546-A1 Abuse-proffed dosage form ENDO PHARMACEUTICALS, INC. 2005-02-10 US disclosed