Dihydromorphine

Dihydromorphine

SCHEMBL13380388

CN1CC[C@]23c4c5ccc(O)c4O[C@H]2[C@@H](O)CCC3C1C5

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 7/20 0.71
OPRK1 P41145 6/20 0.71
OPRM1 P35372 6/20 0.71
MRGPRX2 Q96LB1 2/20 0.64
SLC22A1 O15245 1/20 0.64
ADRA2A P08913 1/20 0.64
ARRB1 P49407 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dihydromorphine SCHEMBL12402795 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL2696539 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL29394226 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL19107002 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL13348852 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL26346 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL19645038 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL19615483 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL17025853 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1
Dihydromorphine SCHEMBL15449768 1.00 OPRD1 (0.71) OPRD1OPRK1OPRM1MRGPRX2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8524904-B2 Process for the preparation of 6-alpha-hydroxy-N-alkylated opiates MALLINCKRODT LLC (US) 2013-09-03 US disclosed
US-8524904-B2 Process for the preparation of 6-alpha-hydroxy-N-alkylated opiates MALLINCKRODT LLC (US) 2013-09-03 US disclosed
US-20100081818-A1 Process for the Preparation of 6-Alpha-Hydroxy-N-Alkylated Opiates MALLINCKRODT INC. (US) 2010-04-01 US disclosed
US-20100081818-A1 Process for the Preparation of 6-Alpha-Hydroxy-N-Alkylated Opiates MALLINCKRODT INC. (US) 2010-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100081818-A1 Process for the Preparation of 6-Alpha-Hydroxy-N-Alkylated Opiates OPRM1, OPRD1, OPRK1 OPRD1 2/4885OPRK1 3/4885OPRM1 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.