SCHEMBL2701145

SCHEMBL2701145

COc1ccccc1N1CCN(C(=O)c2ccc(NS(=O)(=O)c3cccc4cccnc34)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PKM P14618 5/20 1.00
PKLR P30613 16/20 0.75
ALDH1A1 P00352 1/20 0.65
MAPT P10636 1/20 0.65
HTT P42858 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2702266 0.97 PKM (0.93) PKMPKLRALDH1A1MAPTHTT
SCHEMBL12597817 0.91 PKM (0.84) PKMPKLRALDH1A1MAPTHTT
SCHEMBL2704760 0.91 PKM (0.84) PKMPKLR
SCHEMBL2703859 0.91 PKM (0.84) PKMPKLR
SCHEMBL2703998 0.91 PKM (0.83) PKMPKLR
SCHEMBL18753726 0.90 PKM (0.82) PKMPKLR
SCHEMBL2701376 0.90 PKM (0.81) PKMPKLR
SCHEMBL12977013 0.90 PKM (0.81) PKMPKLRALDH1A1MAPTHTT
SCHEMBL2704163 0.90 PKM (0.81) PKMPKLRALDH1A1
SCHEMBL2706093 0.89 PKM (0.80) PKMPKLRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12428376-B2 Therapeutic compounds and compositions AGIOS PHARMACEUTICALS, INC. (US) 2025-09-30 US disclosed
US-20240360083-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS, INC. 2024-10-31 US disclosed
US-11866411-B2 Therapeutic compounds and compositions Agios Pharmaceutical, Inc. (US) 2024-01-09 US disclosed
US-RE49582-E1 Therapeutic compounds and compositions AGIOS PHARMACEUTICALS, INC. (US) 2023-07-18 US disclosed
US-RE49582-E1 Therapeutic compounds and compositions AGIOS PHARMACEUTICALS, INC. (US) 2023-07-18 US disclosed
US-RE49582-E1 Therapeutic compounds and compositions AGIOS PHARMACEUTICALS, INC. (US) 2023-07-18 US disclosed
US-20210198206-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS, INC. 2021-07-01 US disclosed
US-20210198206-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS, INC. 2021-07-01 US disclosed
US-10988448-B2 Therapeutic compounds and compositions AGIOS PHARMACEUTICALS, INC. (US) 2021-04-27 US disclosed
US-10988448-B2 Therapeutic compounds and compositions AGIOS PHARMACEUTICALS, INC. (US) 2021-04-27 US disclosed
US-8785450-B2 Therapeutic compounds and compositions AGIOS PHARMACEUTICALS, INC. (US) 2014-07-22 US disclosed
US-8785450-B2 Therapeutic compounds and compositions AGIOS PHARMACEUTICALS, INC. (US) 2014-07-22 US disclosed
WO-2013056153-A1 ACTIVATORS OF PYRUVATE KINASE M2 AND METHODS OF TREATING DISEASE KUNG CHARLES (US) 2013-04-18 WO disclosed
CN-102481300-A Therapeutic compounds and compositions AGIOS PHARMACEUTICALS INC 2012-05-30 CN disclosed
EP-2448582-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS Agios Pharmaceuticals, Inc. (US) 2012-05-09 EP disclosed
WO-2011002817-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS, INC. (US) 2011-01-06 WO disclosed
WO-2011002817-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS, INC. (US) 2011-01-06 WO disclosed
US-20100331307-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS, INC. 2010-12-30 US disclosed
US-20100331307-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS, INC. 2010-12-30 US disclosed
US-20100331307-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AGIOS PHARMACEUTICALS, INC. 2010-12-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10988448-B2 Therapeutic compounds and compositions PDK1, PDK2, PDK3 PKM 6/4885PKLR 23/4885ALDH1A1 1326/4885
US-20210198206-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS PDK1, PDK2, PDK3 PKM 6/4885PKLR 23/4885ALDH1A1 1326/4885
US-12428376-B2 Therapeutic compounds and compositions PDK1, PDK2, PDK3 PKM 6/4885PKLR 23/4885ALDH1A1 1326/4885
US-20240360083-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS PDK1, PDK2, PDK3 PKM 6/4885PKLR 23/4885ALDH1A1 1326/4885
US-20100331307-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS PDK1, PDK2, PDK3 PKM 6/4885PKLR 23/4885ALDH1A1 1326/4885
US-11866411-B2 Therapeutic compounds and compositions PDK1, PDK2, PDK3 PKM 6/4885PKLR 23/4885ALDH1A1 1326/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.