SCHEMBL2707760

SCHEMBL2707760

Cc1sc([C@@H]2C[C@@H](F)CN2)cc1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
DAO P14920 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSC P53634 1/20 0.31
MAOA P21397 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2136387 0.76 AHR (0.42) ALDH1A1MAOA
SCHEMBL2707575 0.74 PRKAB2 (0.38) MEN1MAPTKMT2A
SCHEMBL2136123 0.66 DPP4 (0.30)
SCHEMBL2708087 0.65 DPP4 (0.44)
SCHEMBL10397862 0.64 ALDH1A1 (0.48) KDM4EMEN1ALDH1A1MAPTDAO
SCHEMBL287087 0.62 ALDH1A1 (0.57) KDM4EMEN1ALDH1A1MAPTDAO
SCHEMBL2724717 0.61 NPC1 (0.37) ALDH1A1
SCHEMBL23633781 0.59 CHRNA1 (0.33)
SCHEMBL18863638 0.59 CHRNA1 (0.33)
SCHEMBL20520605 0.59 KDM4E (0.44) KDM4EMEN1ALDH1A1MAPTDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2447265-A1 NOVEL THIOPHENE CARBOXAMIDE DERIVATIVE AND MEDICINAL USE OF SAME Sanwa Kagaku Kenkyusho Co., Ltd (JP) 2012-05-02 EP disclosed