SCHEMBL27100883

SCHEMBL27100883

CCOC(=O)Nc1sc2c(F)cc(F)c(Br)c2c1C#N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43
BRAF P15056 2/20 0.39
HSD17B10 Q99714 3/20 0.39
RXFP1 Q9HBX9 1/20 0.39
MAPT P10636 5/20 0.38
HPGD P15428 4/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
KDM4E B2RXH2 2/20 0.38
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
TP53 P04637 2/20 0.38
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30781859 1.00 ALDH1A1 (0.47) ALDH1A1NPC1RAB9AALOX15MAPK1
SCHEMBL27147311 0.85 ALDH1A1 (0.38) ALDH1A1NPC1RAB9AMAPK1HSD17B10
SCHEMBL30781872 0.84 TRPA1 (0.35) ALDH1A1NPC1RAB9AALOX15MAPK1
SCHEMBL27100884 0.84 TRPA1 (0.35) ALDH1A1NPC1RAB9AALOX15MAPK1
SCHEMBL29813201 0.84 ALDH1A1 (0.47) ALDH1A1NPC1RAB9AALOX15MAPK1
SCHEMBL23496853 0.84 ALDH1A1 (0.47) ALDH1A1NPC1RAB9AALOX15MAPK1
SCHEMBL31387734 0.84 SMN1; SMN2 (0.40) NPC1RAB9AMAPTPOLBTP53
SCHEMBL24718536 0.77 ALDH1A1 (0.52) ALDH1A1NPC1RAB9AALOX15MAPK1
SCHEMBL25643115 0.75 ALDH1A1 (0.47) ALDH1A1NPC1RAB9AALOX15MAPK1
SCHEMBL30587281 0.74 ALDH1A1 (0.48) ALDH1A1NPC1RAB9AALOX15MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024044667-A2 SMALL MOLECULE INHIBITORS OF KRAS PROTEINS MERCK SHARP & DOHME LLC (US) 2024-02-29 WO disclosed