Lufenuron

Lufenuron

SCHEMBL27105

O=C(NC(=O)c1c(F)cccc1F)Nc1cc(Cl)c(OC(F)(F)C(F)C(F)(F)F)cc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 1.00
MEN1 O00255 4/20 1.00
MAPT P10636 2/20 1.00
USP2 O75604 1/20 1.00
ALOX15 P16050 1/20 1.00
POLB P06746 1/20 0.49
ATM Q13315 1/20 0.46
RECQL P46063 2/20 0.41
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
TLR7 Q9NYK1 1/20 0.38
GAA P10253 2/20 0.38
THRB P10828 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PYGL P06737 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
DHODH Q02127 1/20 0.37
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
IL2 P60568 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lufenuron SCHEMBL4131569 1.00 KMT2A (1.00) KMT2AMEN1MAPTUSP2ALOX15
Lufenuron SCHEMBL29850969 1.00 KMT2A (1.00) KMT2AMEN1MAPTUSP2ALOX15
Lufenuron SCHEMBL15555900 1.00 KMT2A (1.00) KMT2AMEN1MAPTUSP2ALOX15
Lufenuron SCHEMBL28709254 1.00 KMT2A (1.00) KMT2AMEN1MAPTUSP2ALOX15
Lufenuron SCHEMBL29350147 1.00 KMT2A (1.00) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL7587434 0.94 KMT2A (0.88) KMT2AMEN1MAPTUSP2ALOX15
Lufenuron SCHEMBL9990506 0.93 KMT2A (0.87) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL7591855 0.92 KMT2A (0.85) KMT2AMEN1MAPTUSP2ALOX15
Lufenuron SCHEMBL19643246 0.91 MEN1 (0.83) KMT2AMEN1MAPTUSP2ALOX15
SCHEMBL7585954 0.91 KMT2A (0.83) KMT2AMEN1MAPTUSP2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 27861 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137087-A1 INSECTICIDAL COMPOSITIONS RESISTANT TO ACTIVE INGREDIENT DEGRADATION AND PROCESS FOR PREPARATION THEREOF UPL LTD (IN) 2026-05-21 US claimed
CN-122036637-A Polymorphs 先正达农作物保护股份公司 2026-05-15 CN claimed
EP-4734762-A1 BAIT COMPOSITIONS FMC Corporation (US) 2026-05-06 EP claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4723893-A2 COMPOSITIONS AND METHODS TO MITIGATE PHYTOTOXIC EFFECTS OF AGRICHEMICALS Ascribe Bioscience Inc. (US) 2026-04-15 EP claimed
EP-4719059-A1 INCREASED PALATABILITY OF INSECTICIDAL INSECT BAITS Bio Logic Crop Science, S.L. (ES) 2026-04-08 EP claimed
US-20260083129-A1 PYRAZOLE AMIDE INSECTICIDES FMC CORP (US) 2026-03-26 US claimed
US-20260083130-A1 NOVEL SULFONATE BENZAMIDE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS FMC CORP (US) 2026-03-26 US claimed
EP-4709163-A1 MIXTURE COMBINATIONS FOR CROP PROTECTION ADAMA MAKHTESHIM LTD. (IL) 2026-03-18 EP claimed
EP-4709166-A1 NOVEL INSECTICIDAL MIXTURES FOR CONTROLLING AND PROTECTING CROPS ADAMA MAKHTESHIM LTD. (IL) 2026-03-18 EP claimed
WO-1997006687-A1 ACTIVE SUBSTANCE COMBINATIONS COMPRISING PYRETHROIDS AND INSECT-DEVELOPMENT INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 1997-02-27 WO claimed
WO-1996037105-A1 INSECTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-11-28 WO claimed
US-5567429-A PESTICIDES COMPRISING AT LEAST ONE INSECT GROWTH REGULATOR POLYFLUOROPHENYL-ACYLUREA COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-10-22 US claimed
WO-1996029073-A1 NODULISPORIC ACID DERIVATIVES MERCK & CO., INC. (US) 1996-09-26 WO claimed
WO-1996025852-A1 COMPOSITION FOR CONTROLLING PARASITES NOVARTIS AG (CH) 1996-08-29 WO claimed
WO-1995033380-A1 SYNERGISTIC COMPOSITION CIBA-GEIGY AG (CH) 1995-12-14 WO claimed
US-5416102-A Administering orally, by injection or implantation, a dosage of flea growth inhibiting benzoyl urea compound CIBA-GEIGY CORPORATION (US) 1995-05-16 US claimed
WO-1994003066-A1 METHOD AND COMPOSITION FOR CONTROLLING COCKROACHES CIBA-GEIGY AG (CH) 1994-02-17 WO claimed
EP-0518821-A2 Bait station SANDOZ LTD. (CH) 1992-12-16 EP claimed
EP-0433909-A2 Formulation CIBA-GEIGY AG (CH) 1991-06-26 EP claimed