Proglumetacin

Proglumetacin

SCHEMBL27106

CCCN(CCC)C(=O)C(CCC(=O)OCCCN1CCN(CCOC(=O)Cc2c(C)n(C(=O)c3ccc(Cl)cc3)c3ccc(OC)cc23)CC1)NC(=O)c1ccccc1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.59
HTR1A P08908 1/20 0.51
PKM P14618 1/20 0.51
PTGS1 P23219 1/20 0.51
GLO1 Q04760 1/20 0.51
HIF1A Q16665 1/20 0.51
CNR2 P34972 1/20 0.50
AKR1C3 P42330 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Proglumetacin SCHEMBL29384391 1.00 PTGS2 (0.59) PTGS2HTR1APKMPTGS1GLO1
Proglumetacin SCHEMBL19642980 0.97 PTGS2 (0.56) PTGS2HTR1APKMPTGS1GLO1
Proglumetacin SCHEMBL1650599 0.97 PTGS2 (0.56) PTGS2HTR1APKMPTGS1GLO1
Proglumetacin SCHEMBL99165 0.97 PTGS2 (0.56) PTGS2HTR1APKMPTGS1GLO1
Proglumetacin SCHEMBL2070226 0.97 PTGS2 (0.55) PTGS2PTGS1
Proglumetacin SCHEMBL28086382 0.97 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL5077578 0.91 PTGS2 (0.57) PTGS2HTR1APKMPTGS1GLO1
Proglumetacin SCHEMBL4094289 0.91 PTGS2 (0.52) PTGS2
Proglumetacin SCHEMBL13724384 0.91 PTGS2 (0.49) PTGS2HTR1APKMPTGS1GLO1
Proglumetacin SCHEMBL5482765 0.89 PTGS2 (0.47) PTGS2HTR1APKMPTGS1GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4877 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ACERAGEN INC (US) 2026-01-01 US claimed
US-20250041208-A1 NEW INJECTABLE COMBINATION FORMULATION NANEXA AB (SE) 2025-02-06 US claimed
EP-3508501-B1 USE OF ANTI-CGRP ANTIBODIES AND ANTIBODY FRAGMENTS TO PREVENT OR INHIBIT PHOTOPHOBIA OR LIGHT AVERSION IN SUBJECTS IN NEED THEREOF, ESPECIALLY MIGRAINE SUFFERERS H LUNDBECK AS (DK) 2024-11-06 EP claimed
EP-4444277-A1 NEW INJECTABLE COMBINATION FORMULATION Nanexa AB (SE) 2024-10-16 EP claimed
WO-2024105529-A1 CHEMICAL DISBUDDING OF LIVESTOCK MASSEY UNIVERSITY (NZ) 2024-05-23 WO claimed
EP-4340884-A1 TREATMENT OF INFECTIONS IN AND AROUND THE EYE University of Miami (US) 2024-03-27 EP claimed
WO-2024027794-A1 TASTE-MASKING MICROSPHERE, PREPARATION PROCESS THEREFOR, AND USE THEREOF 哈尔滨市康隆药业有限责任公司 2024-02-08 WO claimed
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
WO-2023105227-A1 NEW INJECTABLE COMBINATION FORMULATION NANEXA AB (SE) 2023-06-15 WO claimed
WO-2022245950-A1 TREATMENT OF INFECTIONS IN AND AROUND THE EYE UNIVERSITY OF MIAMI (US) 2022-11-24 WO claimed
US-5818002-A Pressure change warning switch CTS CORPORATION (US) 1998-10-06 US claimed
EP-0759750-A4 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1998-05-27 EP claimed
WO-1997037680-A1 MACROMOLECULAR COMPLEXES FOR DRUG DELIVERY THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1997-10-16 WO claimed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP claimed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP claimed
EP-0759750-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO, Howard, K. (US) 1997-03-05 EP claimed
US-5543417-A 5 Alpha-reductase inhibitor and at least one of an antibacterial agent, a keratolytic agent or an anti-inflammatory agent MERCK & CO., INC. (US) 1996-08-06 US claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1995031194-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1995-11-23 WO claimed