SCHEMBL27140362

SCHEMBL27140362

CCOCc1cnc(Cl)nc1N

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.45
CSNK1A1 P48729 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
DHFR P00374 2/20 0.38
CGAS Q8N884 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17581276 0.82 KDM4E (0.33)
SCHEMBL11396782 0.82 DHFR (0.54) DHFR
SCHEMBL22895290 0.81 KDM4E (0.32)
SCHEMBL7724215 0.81 LMNA (0.69) LMNA
SCHEMBL27153028 0.77 ALDH1A1 (0.36) LMNA
SCHEMBL30891184 0.77 ALDH1A1 (0.36) LMNA
SCHEMBL21593668 0.77 CSNK1A1 (0.43) LMNACSNK1A1CLK4DHFR
SCHEMBL25323208 0.73 TLR8 (0.45) CSNK1A1CLK4
SCHEMBL30068026 0.73 TLR8 (0.45) CSNK1A1CLK4
SCHEMBL30042167 0.72 TLR8 (0.46) CSNK1A1CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024044731-A1 DIAZEPINO-THIENO-QUINOXALINE COMPOUNDS AND THEIR USE IN THERAPY MATCHPOINT THERAPEUTICS INC. (US) 2024-02-29 WO disclosed
WO-2024044731-A1 DIAZEPINO-THIENO-QUINOXALINE COMPOUNDS AND THEIR USE IN THERAPY MATCHPOINT THERAPEUTICS INC. (US) 2024-02-29 WO disclosed