SCHEMBL2714877

SCHEMBL2714877

CCN(C(=O)C1(C(N)=O)CC1)c1ccc(Br)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.47
RAB9A P51151 5/20 0.36
NPC1 O15118 3/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KMT2A Q03164 1/20 0.35
OPRK1 P41145 1/20 0.34
ADRA2A P08913 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
PLAU P00749 1/20 0.34
FPR2 P25090 1/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPK1 P28482 1/20 0.32
TSHR P16473 1/20 0.32
RXRA P19793 2/20 0.32
RXRB P28702 2/20 0.32
RXRG P48443 2/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2713483 0.77 OXTR (0.35) ALDH1A1OPRK1FPR2TSHR
SCHEMBL856442 0.73 GBA1 (0.48) GBA1RAB9ANPC1ALDH1A1MAPT
SCHEMBL24100191 0.71 GBA1 (0.53) GBA1RAB9ANPC1ALDH1A1MAPT
SCHEMBL1180593 0.69 GBA1 (0.50) GBA1RAB9ANPC1ALDH1A1MAPT
SCHEMBL19260095 0.67 GBA1 (0.43) GBA1RAB9ANPC1ALDH1A1MAPT
SCHEMBL2714876 0.67 FPR2 (0.44) RAB9ANPC1ALDH1A1SMN1; SMN2KMT2A
SCHEMBL17316578 0.65 GBA1 (1.00) GBA1RAB9ANPC1ALDH1A1MAPT
SCHEMBL18988815 0.65 GBA1 (0.42) GBA1RAB9ANPC1ALDH1A1MAPT
SCHEMBL20742815 0.65 USP30 (0.50) GBA1RAB9ANPC1ALDH1A1MAPT
SCHEMBL20742814 0.65 USP30 (0.50) GBA1RAB9ANPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445909-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-a]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES Boehringer Ingelheim International GmbH (DE) 2012-05-02 EP disclosed
WO-2010141273-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-a]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-09 WO disclosed