Revizinone

Revizinone

SCHEMBL27163

CN(C(=O)CO/N=C(\c1ccccc1)c1ccc2c(c1)CN1CC(=O)N=C1N2)C1CCCCC1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 19/20 0.50
PDE3A Q14432 19/20 0.50
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
P2RY12 Q9H244 1/20 0.45
BACE1 P56817 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Revizinone SCHEMBL9584593 0.87 PDE3B (0.68) PDE3BPDE3APDE4APDE4BPDE4C
Revizinone SCHEMBL7297062 0.87 PDE3B (0.68) PDE3BPDE3APDE4APDE4BPDE4C
Revizinone SCHEMBL29557974 0.87 PDE3B (0.68) PDE3BPDE3APDE4APDE4BPDE4C
Revizinone SCHEMBL7289525 0.87 PDE3B (0.68) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9583372 0.78 PDE3B (0.70) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9584441 0.78 PDE3B (0.70) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9583358 0.78 PDE3B (0.70) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9584335 0.78 PDE3B (0.72) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9584347 0.78 PDE3B (0.72) PDE3BPDE3APDE4APDE4BPDE4C
Water SCHEMBL9583863 0.78 PDE3B (0.71) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 778 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023196821-A2 TARGETING NEUROPOD CELL GUCY2C TO CONTROL VISCERAL PAIN AND APPETITE THOMAS JEFFERSON UNIVERSITY (US) 2023-10-12 WO claimed
EP-3532008-A1 TREATMENT OF GYNOID LIPODYSTROPHY Merz Pharma GmbH & Co. KGaA (DE) 2019-09-04 EP claimed
WO-2019164836-A1 SYSTEMS AND METHODS FOR COMBINED COSMETIC TREATMENT OF CELLULITE WITH ULTRASOUND ULTHERA, INC. (US) 2019-08-29 WO claimed
US-20190240253-A1 TREATMENT OF GYNOID LIPODYSTROPHY MERZ PHARMA GMBH & CO. KGAA (DE) 2019-08-08 US claimed
WO-2018077825-A1 TREATMENT OF GYNOID LIPODYSTROPHY MERZ PHARMA GMBH & CO. KGAA (DE) 2018-05-03 WO claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20050130971-A1 Compositions of a cyclooxygenase-2 selective inhibitor and phosphodiesterase inhibitor for the treatment of ischemic mediated central nervous system disorders or injury PHARMACIA CORPORATION 2005-06-16 US claimed
WO-2005018563-A2 COMPOSITIONS OF A CYCLOOXYGENASE-2 SELECTIVE INHIBITOR AND A PHOSPHODIESTERASE INHIBITOR FOR THE TREATMENT OF ISCHEMIC MEDIATED CENTRAL NERVOUS SYSTEM DISORDERS OR INJURY PHARMACIA CORPORATION (US) 2005-03-03 WO claimed
EP-1370211-A4 CO-ADMINISTRATION OF MELANOCORTIN RECEPTOR AGONIST AND PHOSPHODIESTERASE INHIBITOR FOR TREATMENT OF CYCLIC-AMP ASSOCIATED DISORDERS BRISTOL MYERS SQUIBB CO (US) 2005-02-09 EP claimed
EP-1370211-A2 CO-ADMINISTRATION OF MELANOCORTIN RECEPTOR AGONIST AND PHOSPHODIESTERASE INHIBITOR FOR TREATMENT OF CYCLIC-AMP ASSOCIATED DISORDERS Bristol-Myers Squibb Company (US) 2003-12-17 EP claimed
US-20030069169-A1 Co-administration of melanocortin receptor agonist and phosphodiesterase inhibitor for treatment of cyclic-AMP associated disorders BRISTOL-MYERS SQUIBB COMPANY 2003-04-10 US claimed
WO-2002069905-A2 CO-ADMINISTRATION OF MELANOCORTIN RECEPTOR AGONIST AND PHOSPHODIESTERASE INHIBITOR FOR TREATMENT OF CYCLIC-AMP ASSOCIATED DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2002-09-12 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190240253-A1 TREATMENT OF GYNOID LIPODYSTROPHY FABP4, GYS1, EBP PDE3B 3564/4885PDE3A 3100/4885PDE4A 2435/4885
US-20030069169-A1 Co-administration of melanocortin receptor agonist and phosphodiesterase inhibitor for treatment of cyclic-AMP associated disorders MC4R, MC3R, MC1R PDE3B 66/4885PDE3A 88/4885PDE4A 6/4885
US-20050130971-A1 Compositions of a cyclooxygenase-2 selective inhibitor and phosphodiesterase inhibitor for the treatment of ischemic mediated central nervous system disorders or injury PDE2A, PDE3B, PDE3A PDE3B 2/4885PDE3A 3/4885PDE4A 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.