SCHEMBL27163155

SCHEMBL27163155

O=C1C(=O)N(C2CCCC2)CCN1Cc1ccc(Cl)nc1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.54
ALDH1A1 P00352 1/20 0.51
GRM2 Q14416 1/20 0.47
IL4I1 Q96RQ9 1/20 0.47
CHRNA1 P02708 1/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA7 P36544 1/20 0.47
CHRNA4 P43681 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30947906 0.84 TP53 (0.48) TP53IL4I1LMNA
SCHEMBL27163372 0.83 TP53 (0.47) TP53IL4I1LMNA
SCHEMBL27163582 0.82 IL4I1 (0.62) TP53IL4I1LMNA
SCHEMBL30046438 0.82 IL4I1 (0.62) TP53IL4I1LMNA
SCHEMBL30948336 0.82 IL4I1 (0.47) TP53IL4I1LMNA
SCHEMBL30948316 0.81 TP53 (0.47) TP53IL4I1LMNA
SCHEMBL30948055 0.80 TP53 (0.54) TP53IL4I1LMNA
SCHEMBL30947968 0.80 IL4I1 (0.49) TP53IL4I1LMNA
SCHEMBL30948110 0.79 TP53 (0.47) TP53IL4I1LMNA
SCHEMBL30948268 0.79 TP53 (0.44) TP53IL4I1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240246937-A1 IL4I1 INHIBITORS AND METHODS OF USE MERCK SHARP & DOHME LLC (US) 2024-07-25 US disclosed
EP-4329889-A1 IL4I1 INHIBITORS AND METHODS OF USE Merck Sharp & Dohme LLC (US) 2024-03-06 EP disclosed
WO-2022227015-A1 IL4I1 INHIBITORS AND METHODS OF USE MERCK SHARP & DOHME CORP. (US) 2022-11-03 WO disclosed
WO-2022232333-A1 IL4I1 INHIBITORS AND METHODS OF USE MERCK SHARP & DOHME LLC (US) 2022-11-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240246937-A1 IL4I1 INHIBITORS AND METHODS OF USE IL4I1, IL4, IL2 TP53 1444/4885ALDH1A1 283/4885GRM2 4617/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.