SCHEMBL2719948

SCHEMBL2719948

O=C(O)NCCc1nc2ccc(F)cc2c(CO)c1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
DHODH Q02127 9/20 0.46
PRNP P04156 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
PLA2G2A P14555 2/20 0.40
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
TACR1 P25103 1/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
PRKAA2 P54646 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2718169 0.86 ALDH1A1 (0.45) ALDH1A1DHODHPRNPTDP1PLA2G2A
SCHEMBL2717623 0.86 CKS1B (0.41) ALDH1A1DHODHPRNPTDP1PLA2G2A
SCHEMBL2717984 0.82 DHODH (0.50) ALDH1A1DHODHPRNPTDP1POLB
SCHEMBL6122794 0.78 ALDH1A1 (0.47) ALDH1A1DHODHPLA2G2AMAPTMEN1
SCHEMBL2719964 0.76 ALDH1A1 (0.45) ALDH1A1TDP1PLA2G2APOLBMAPT
SCHEMBL2717553 0.76 IDO1 (0.40) ALDH1A1DHODHPRNPPLA2G2APOLB
SCHEMBL2719179 0.75 GNRHR (0.42) ALDH1A1DHODHPRNPMTNR1AMTNR1B
SCHEMBL3784083 0.75 DHODH (0.47) ALDH1A1DHODHPRNPTDP1PLA2G2A
SCHEMBL2717125 0.74 PIK3CD (0.57)
SCHEMBL2717794 0.74 GNRHR (0.41) ALDH1A1DHODHPRNPPLA2G2AMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445900-A2 POLYCYCLIC DERIVATIVES OF PYRIDINE AND THEIR USE IN THE TREATMENT OF (INTER ALIA) RHEUMATOID ARTHRITIS AND SIMILAR DISEASES Amgen, Inc (US) 2012-05-02 EP disclosed
WO-2010151740-A2 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2010-12-29 WO disclosed