SCHEMBL2719964

SCHEMBL2719964

O=C(O)NCCc1nc2ccc(F)cc2c(Cl)c1-c1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
PIK3CD O00329 3/20 0.43
PIK3CA P42336 3/20 0.43
PIK3CB P42338 3/20 0.43
PIK3CG P48736 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.40
NAMPT P43490 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
PLA2G2A P14555 1/20 0.39
P2RX7 Q99572 1/20 0.39
CTSD P07339 1/20 0.38
GUSB P08236 1/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
AGTR1 P30556 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6122794 0.91 ALDH1A1 (0.47) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2717092 0.86 GNRHR (0.41) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2716683 0.86 PIK3CD (0.46) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL6122682 0.84 PIK3CD (0.48) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL6122848 0.83 ALDH1A1 (0.44) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2718718 0.82 PIK3CD (0.47) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2718336 0.79 PIK3CD (0.48) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL6128776 0.78 ALDH1A1 (0.41) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2719948 0.76 ALDH1A1 (0.47) ALDH1A1HPGDPLA2G2APOLBMAPT
SCHEMBL2718042 0.76 PIK3CD (0.40) ALDH1A1PIK3CDPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445900-A2 POLYCYCLIC DERIVATIVES OF PYRIDINE AND THEIR USE IN THE TREATMENT OF (INTER ALIA) RHEUMATOID ARTHRITIS AND SIMILAR DISEASES Amgen, Inc (US) 2012-05-02 EP disclosed
WO-2010151740-A2 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2010-12-29 WO disclosed