SCHEMBL2720103

SCHEMBL2720103

CCCC[C@](C)(N)C(=O)O.CSCC[C@](C)(N)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ARG1 P05089 2/20 0.47
ARG2 P78540 2/20 0.47
GGT1 P19440 1/20 0.43
FDPS P14324 3/20 0.36
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
NOS3 P29474 1/20 0.35
BLM P54132 3/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP1A2 P05177 2/20 0.33
POLB P06746 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 1/20 0.33
USP2 O75604 1/20 0.33
EGFR P00533 1/20 0.33
FYN P06241 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL162014 0.89 GGT1 (0.52) ARG1ARG2GGT1NOS1NOS2
SCHEMBL5614525 0.89 GGT1 (0.52) ARG1ARG2GGT1NOS1NOS2
SCHEMBL243496 0.89 GGT1 (0.52) ARG1ARG2GGT1NOS1NOS2
SCHEMBL5614536 0.89 GGT1 (0.52) ARG1ARG2GGT1NOS1NOS2
SCHEMBL162368 0.89 GGT1 (0.52) ARG1ARG2GGT1NOS1NOS2
Hydrochloric Acid SCHEMBL13585526 0.87 GGT1 (0.50) ARG1ARG2GGT1NOS1NOS2
SCHEMBL186714 0.87 ARG1 (0.59) ARG1ARG2GGT1FDPSBLM
SCHEMBL18124758 0.87 ARG1 (0.59) ARG1ARG2GGT1FDPSBLM
SCHEMBL162337 0.87 ARG1 (0.59) ARG1ARG2GGT1FDPSBLM
Hydrochloric Acid SCHEMBL18109448 0.85 ARG1 (0.57) ARG1ARG2GGT1FDPSNOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3472192-A1 SPIDER VENOM PEPTIDES AND METHODS OF USE FOR MODULATING SODIUM CHANNELS. The University of Queensland (AU) 2019-04-24 EP disclosed
EP-3411061-A1 PROTEINACEOUS COMPOUNDS AND USES THEREFOR University of Canberra (AU) 2018-12-12 EP disclosed
EP-3387007-A1 PROTEINACEOUS MOLECULES AND METHODS OF USE The University of Queensland (AU) 2018-10-17 EP disclosed
WO-2017219081-A1 SPIDER VENOM PEPTIDES AND METHODS OF USE FOR MODULATING SODIUM CHANNELS. THE UNIVERSITY OF QUEENSLAND (AU) 2017-12-28 WO disclosed
WO-2017132728-A1 PROTEINACEOUS COMPOUNDS AND USES THEREFOR UNIVERSITY OF CANBERRA (AU) 2017-08-10 WO disclosed
WO-2017096431-A1 PROTEINACEOUS MOLECULES AND METHODS OF USE THE UNIVERSITY OF QUEENSLAND (AU) 2017-06-15 WO disclosed
EP-2726154-A1 PREVENTION AND TREATMENT OF ACUTE INFLAMMATORY CONDITIONS The University of Queensland (AU) 2014-05-07 EP disclosed
EP-2681238-A2 APOPTOSIS-INDUCING MOLECULES AND USES THEREFOR Istituto di Ricovero E Cura A Carattere Scientifico Materno-Infantile Burlo Garofolo- Ospedale di Alta Specializzazione E di Rilievo (IT) 2014-01-08 EP disclosed
EP-2635596-A1 IMMUNE-MODULATING AGENTS AND USES THEREFOR UNIVERSITY OF TECHNOLOGY, SYDNEY (AU) 2013-09-11 EP disclosed
WO-2013026105-A1 PEST-CONTROLLING AGENTS ISOLATED FROM SPIDER VENOM AND USES THEREOF THE UNIVERSITY OF QUEENSLAND (AU) 2013-02-28 WO disclosed
WO-2009089568-A1 IMMUNOMODULATING COMPOSITIONS AND USES THEREFOR OPAL THERAPEUTICS PTY LTD (AU) 2009-07-23 WO disclosed
EP-1285004-A4 SYNTHETIC PEPTIDES AND USES THEREFORE UNIV AUSTRALIAN (AU) 2006-03-29 EP disclosed
EP-1078003-A4 PLASMIN INHIBITORS FROM THE AUSTRALIAN BROWN SNAKE $i(PSEUDONAJA TEXTILIS TEXTILIS) UNIV QUEENSLAND (AU) 2004-08-25 EP disclosed
EP-1285004-A1 SYNTHETIC PEPTIDES AND USES THEREFORE THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2003-02-26 EP disclosed
WO-2001090197-A1 SYNTHETIC PEPTIDES AND USES THEREFORE THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2001-11-29 WO disclosed
EP-1045859-A4 NOVEL SURFACE PROTEIN OF $i(NEISSERIA MENINGITIDIS) UNIV QUEENSLAND (AU) 2001-08-22 EP disclosed
EP-1078003-A1 PLASMIN INHIBITORS FROM THE AUSTRALIAN BROWN SNAKE $i(PSEUDONAJA TEXTILIS TEXTILIS) THE UNIVERSITY OF QUEENSLAND (AU) 2001-02-28 EP disclosed
EP-1045859-A1 NOVEL SURFACE PROTEIN OF $i(NEISSERIA MENINGITIDIS) THE UNIVERSITY OF QUEENSLAND (AU) 2000-10-25 EP disclosed
WO-1999058569-A1 PLASMIN INHIBITORS FROM THE AUSTRALIAN BROWN SNAKE $i(PSEUDONAJA TEXTILIS TEXTILIS) THE UNIVERSITY OF QUEENSLAND (AU) 1999-11-18 WO disclosed
WO-1999031132-A1 NOVEL SURFACE PROTEIN OF $i(NEISSERIA MENINGITIDIS) THE UNIVERSITY OF QUEENSLAND (AU) 1999-06-24 WO disclosed