SCHEMBL2720281

SCHEMBL2720281

Cc1c(OC2CCNCC2)ncnc1N1CCc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.43
GPR119 Q8TDV5 14/20 0.39
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
WDR5 P61964 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP2C9 P11712 2/20 0.36
EIF4E P06730 2/20 0.36
MKNK1 Q9BUB5 2/20 0.36
MKNK2 Q9HBH9 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1066161 0.83 GPR119 (0.58) GPR119CYP2C9
SCHEMBL3716443 0.70 GPR119 (0.47) GPR119CYP2C9
SCHEMBL8647897 0.69 EGFR (0.67) HTTSMN1; SMN2
SCHEMBL12236499 0.69 HRH4 (0.43) HTT
SCHEMBL288618 0.69 GPR119 (0.75) GPR119CYP2C9
SCHEMBL16701160 0.68 SMN1; SMN2 (0.45) HTTSMN1; SMN2KMT2A
SCHEMBL12236467 0.68 HRH1 (0.43) GPR119
SCHEMBL761736 0.67 GPR119 (0.58) GPR119CYP2C9
SCHEMBL3304134 0.66 ALDH1A1 (0.54) WDR5KMT2ACYP3A4CYP2C19
SCHEMBL3181260 0.66 ALDH1A1 (0.39) IRAK4HTTSMN1; SMN2KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445901-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO Boehringer Ingelheim International GmbH (DE) 2012-05-02 EP disclosed
WO-2010149685-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-29 WO disclosed