Radezolid

Radezolid

SCHEMBL2723587

CC(=O)NC[C@H]1CN(c2ccc(-c3ccc(CNCc4cnn[nH]4)cc3)c(F)c2)C(=O)O1.Cl

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

rplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Radezolid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.55
CALML3 P27482 7/20 0.50
MAOB P27338 2/20 0.50
LMNA P02545 1/20 0.50
PTGS1 P23219 1/20 0.50
SDHA P31040 1/20 0.50
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Radezolid SCHEMBL1035776 0.99 MAOA (0.56) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL3165892 0.99 MAOA (0.56) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL30061945 0.99 MAOA (0.56) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL15633880 0.98 MAOA (0.55) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL15634852 0.96 MAOA (0.53) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL15634976 0.96 MAOA (0.53) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL15634749 0.95 MAOA (0.52) MAOACALML3MAOBLMNAPTGS1
SCHEMBL12956217 0.93 MAOA (0.54) MAOACALML3MAOBLMNAPTGS1
SCHEMBL1036539 0.93 MAOA (0.54) MAOACALML3MAOBLMNAPTGS1
SCHEMBL1032249 0.93 MAOA (0.54) MAOACALML3MAOBLMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9126991-B2 Radezolid salts and polymorphic forms thereof LI HUI-YIN (US) 2015-09-08 US claimed
US-20140100254-A1 Radezolid salts and polymorphic forms thereof LI HUI-YIN (US) 2014-04-10 US claimed
EP-4184568-B1 HIGH-FREQUENCY PACKAGE NTT INC (JP) 2026-05-13 EP disclosed
US-12489069-B2 High frequency package NTT, INC. (JP) 2025-12-02 US disclosed
EP-4191659-B1 PRODUCTION METHOD FOR HIGH-FREQUENCY PACKAGE NTT INC (JP) 2025-11-05 EP disclosed
EP-4191657-B1 PACKAGE AND PRODUCTION METHOD THEREFOR NTT INC (JP) 2025-10-01 EP disclosed
US-12322668-B2 Package and manufacturing method of the same NIPPON TELEGRAPH AND TELEPHONE CORPORATION (JP) 2025-06-03 US disclosed
US-12272567-B2 Manufacturing method for high-frequency package NIPPON TELEGRAPH AND TELEPHONE CORPORATION (JP) 2025-04-08 US disclosed
US-20240421107-A1 MOUNTING STRUCTURE NTT, INC. (JP) 2024-12-19 US disclosed
EP-4191659-A1 PRODUCTION METHOD FOR HIGH-FREQUENCY PACKAGE NIPPON TELEGRAPH AND TELEPHONE CORPORATION (JP) 2023-06-07 EP disclosed
EP-4191657-A1 PACKAGE AND PRODUCTION METHOD THEREFOR NIPPON TELEGRAPH AND TELEPHONE CORPORATION (JP) 2023-06-07 EP disclosed
EP-3970734-A2 COMPARTMENTALIZED METHOD OF NUCLEIC ACID DELIVERY AND COMPOSITIONS AND USES THEREOF Global Bio Therapeutics, Inc. (US) 2022-03-23 EP disclosed
WO-2022029838-A1 PACKAGE AND PRODUCTION METHOD THEREFOR 日本電信電話株式会社 2022-02-10 WO disclosed
WO-2022024289-A1 PRODUCTION METHOD FOR HIGH-FREQUENCY PACKAGE 日本電信電話株式会社 2022-02-03 WO disclosed
EP-2635307-B1 PHARMACEUTICAL COMPOSITIONS MELINTA SUBSIDIARY CORP (US) 2020-07-29 EP disclosed
US-9409896-B2 Sustained release pharmaceutical compositions comprising an antibacterial agent MELINTA THERAPEUTICS, INC. (US) 2016-08-09 US disclosed
US-9126991-B2 Radezolid salts and polymorphic forms thereof LI HUI-YIN (US) 2015-09-08 US disclosed
US-20140100254-A1 Radezolid salts and polymorphic forms thereof LI HUI-YIN (US) 2014-04-10 US disclosed
EP-2635307-A2 PHARMACEUTICAL COMPOSITIONS Rib-X Pharmaceuticals, Inc. (US) 2013-09-11 EP disclosed
WO-2012061360-A2 PHARMACEUTICAL COMPOSITIONS RIB-X PHARMACEUTICALS, INC. (US) 2012-05-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140100254-A1 Radezolid salts and polymorphic forms thereof RPL27A, GRHPR, RAD52 MAOA 3452/4885CALML3 2920/4885MAOB 2745/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.