Radezolid

Radezolid

SCHEMBL1035776

CC(=O)NC[C@H]1CN(c2ccc(-c3ccc(CNCc4cnn[nH]4)cc3)c(F)c2)C(=O)O1

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

rplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Radezolid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.56
CALML3 P27482 7/20 0.51
MAOB P27338 2/20 0.51
LMNA P02545 1/20 0.51
PTGS1 P23219 1/20 0.51
SDHA P31040 1/20 0.51
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Radezolid SCHEMBL3165892 1.00 MAOA (0.56) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL30061945 1.00 MAOA (0.56) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL15633880 0.99 MAOA (0.55) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL2723587 0.99 MAOA (0.55) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL15634976 0.97 MAOA (0.53) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL15634852 0.97 MAOA (0.53) MAOACALML3MAOBLMNAPTGS1
Radezolid SCHEMBL15634749 0.96 MAOA (0.52) MAOACALML3MAOBLMNAPTGS1
SCHEMBL12956217 0.93 MAOA (0.54) MAOACALML3MAOBLMNAPTGS1
SCHEMBL1032249 0.93 MAOA (0.54) MAOACALML3MAOBLMNAPTGS1
SCHEMBL1036539 0.93 MAOA (0.54) MAOACALML3MAOBLMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1105 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4727950-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE IN THE TREATMENT OF MYCOBACTERIAL INFECTIONS GlaxoSmithKline Intellectual Property Development Ltd (GB) 2026-04-22 EP claimed
US-20260048047-A1 SMALL-MOLECULE ACTIVATORS OF MYCOBACTERIUM TUBERCULOSIS ADENYLYL CYCLASE SCRIPPS RESEARCH INST (US) 2026-02-19 US claimed
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA ATOPIC MEDICAL INC (US) 2026-01-29 US claimed
EP-4027535-B1 WIRELESS TRANSCEIVER DEVICE INTEGRATED WITH COMMON CLOCK PHASE-LOCKED LOOP HUAWEI TECH CO LTD (CN) 2025-12-03 EP claimed
US-12465623-B2 Use of parasites and extracellular vesicles obtained from parasites in cancer treatment YEDITEPE UNIVERSITESI (TR) 2025-11-11 US claimed
EP-3965808-B1 USE OF PARASITES AND EXTRACELLULAR VESICLES OBTAINED FROM PARASITES IN CANCER TREATMENT UNIV YEDITEPE (TR) 2025-09-03 EP claimed
WO-2025096495-A1 ARYL FLUOROSULFATE-BASED INHIBITORS AS NOVEL ANTITUBERCULAR AGENTS THE SCRIPPS RESEARCH INSTITUTE (US) 2025-05-08 WO claimed
US-12285489-B2 Bone targeted antimicrobial oxazolidinone related compounds, formulations thereof, and uses thereof EBETINO FRANK HALLOCK (US) 2025-04-29 US claimed
US-20250129084-A1 Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2025-04-24 US claimed
WO-2025080590-A1 CO-CRYSTALLIZATION OF ACTIVES WITH SACCHARIDE-BASED MOLECULAR FRAMEWORKS SCIENTIFIC HORIZONS CONSULTING LLC (US) 2025-04-17 WO claimed
US-20220170104-A1 BACTERIAL ETIOLOGY OF COLORECTAL CANCER DANA-FARBER CANCER INSTITUTE, INC. 2022-06-02 US claimed
WO-2022114728-A2 COMPOSITION COMPRISING SHMT INHIBITOR OR MTHFR INHIBITOR FOR TREATING BACTERIAL INFECTION 성균관대학교산학협력단 2022-06-02 WO claimed
EP-3965808-A1 USE OF PARASITES AND EXTRACELLULAR VESICLES OBTAINED FROM PARASITES IN CANCER TREATMENT Yeditepe Universitesi (TR) 2022-03-16 EP claimed
US-11248259-B2 Method of identifying a subject having a bacterial infection IMPERIAL COLLEGE OF SCIENCE, TECHNOLOGY AND MEDICINE (GB) 2022-02-15 US claimed
EP-2635307-B1 PHARMACEUTICAL COMPOSITIONS MELINTA SUBSIDIARY CORP (US) 2020-07-29 EP claimed
US-9409896-B2 Sustained release pharmaceutical compositions comprising an antibacterial agent MELINTA THERAPEUTICS, INC. (US) 2016-08-09 US claimed
US-9126991-B2 Radezolid salts and polymorphic forms thereof LI HUI-YIN (US) 2015-09-08 US claimed
US-20140100254-A1 Radezolid salts and polymorphic forms thereof LI HUI-YIN (US) 2014-04-10 US claimed
EP-2635307-A2 PHARMACEUTICAL COMPOSITIONS Rib-X Pharmaceuticals, Inc. (US) 2013-09-11 EP claimed
WO-2012061360-A2 PHARMACEUTICAL COMPOSITIONS RIB-X PHARMACEUTICALS, INC. (US) 2012-05-10 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA IL1B, IL5, SERPINB1 MAOA 416/4885CALML3 1297/4885MAOB 46/4885
US-20250129084-A1 Compounds CFTR, TBCA, TBCD MAOA 2138/4885CALML3 2453/4885MAOB 1545/4885
US-20140100254-A1 Radezolid salts and polymorphic forms thereof RPL27A, GRHPR, RAD52 MAOA 3452/4885CALML3 2920/4885MAOB 2745/4885
US-20260048047-A1 SMALL-MOLECULE ACTIVATORS OF MYCOBACTERIUM TUBERCULOSIS ADENYLYL CYCLASE FNTB, PDE7A, TBL3 MAOA 1993/4885CALML3 1019/4885MAOB 1339/4885
US-12285489-B2 Bone targeted antimicrobial oxazolidinone related compounds, formulations thereof, and uses thereof SOST, BPGM, PTMS MAOA 3576/4885CALML3 4370/4885MAOB 2694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.