SCHEMBL27248697

SCHEMBL27248697

COCCOc1cccc2nc(O)nc(O)c12

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 8/20 0.44
TSHR P16473 1/20 0.41
KDM1A O60341 1/20 0.39
EGFR P00533 1/20 0.37
DCPS Q96C86 3/20 0.36
DHFR P00374 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
CYBB P04839 1/20 0.35
NOX5 Q96PH1 1/20 0.35
JAK2 O60674 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
FGFR1 P11362 1/20 0.35
FLT1 P17948 1/20 0.35
MIF P14174 1/20 0.35
IKBKB O14920 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16011941 0.81 ALDH1A1 (0.53) TSHRDCPSDHFRKDM4EALDH1A1
SCHEMBL1192087 0.81 EGFR (0.45) NCF1TSHRKDM1AEGFRJAK2
SCHEMBL27248729 0.74 TLR8 (0.40) TSHRDCPSDHFRKDM4EALDH1A1
SCHEMBL27248810 0.73 NCF1 (0.44) NCF1TSHRKDM1ADCPSDHFR
SCHEMBL1154579 0.73 DCPS (0.68) NCF1DCPSDHFR
SCHEMBL3402989 0.72 DCPS (0.50) NCF1DCPSDHFR
SCHEMBL29041258 0.72 NCF1 (0.52) NCF1TSHRDCPSDHFRCYBB
SCHEMBL27248935 0.71 KCNH2 (0.38) DCPSKDM4EALDH1A1HPGDMAPT
SCHEMBL3686238 0.70 NCF1 (0.49) NCF1TSHRKDM1AEGFRKDM4E
SCHEMBL1192699 0.69 KDM1A (0.45) NCF1TSHRKDM1AEGFRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240360085-A1 Glucose Uptake Inhibitors KADMON CORPORATION, LLC (US) 2024-10-31 US disclosed
US-12030857-B2 Glucose uptake inhibitors KADMON CORPORATION, LLC (US) 2024-07-09 US disclosed
US-12030857-B2 Glucose uptake inhibitors KADMON CORPORATION, LLC (US) 2024-07-09 US disclosed
US-12030857-B2 Glucose uptake inhibitors KADMON CORPORATION, LLC (US) 2024-07-09 US disclosed
US-20220363648-A1 Glucose Uptake Inhibitors KADMON CORPORATION, LLC 2022-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12030857-B2 Glucose uptake inhibitors SLC2A1, SLC2A4, SLC2A2 NCF1 1313/4885TSHR 3168/4885KDM1A 2270/4885
US-20220363648-A1 Glucose Uptake Inhibitors SLC2A1, SLC2A4, SLC2A2 NCF1 1313/4885TSHR 3168/4885KDM1A 2270/4885
US-20240360085-A1 Glucose Uptake Inhibitors SLC2A3, SLC2A1, SLC2A4 NCF1 1399/4885TSHR 2854/4885KDM1A 1991/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.