SCHEMBL27263162

SCHEMBL27263162

Fc1ccc(F)cc1.O=CCl

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
ACHE P22303 1/20 0.42
HSD11B1 P28845 2/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
NFE2L2 Q16236 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
FBP1 P09467 1/20 0.37
IDO1 P14902 1/20 0.36
ORAI1 Q96D31 1/20 0.36
ORAI2 Q96SN7 1/20 0.36
ORAI3 Q9BRQ5 1/20 0.36
TRPV6 Q9H1D0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27427610 0.86 APP (0.42) CES2CES1CA1CA2CA7
SCHEMBL27372250 0.86 ACHE (0.68) ACHELMNANFE2L2
SCHEMBL27882939 0.86 SMN1; SMN2 (0.43) CES2CES1HSD11B1ALDH1A1LMNA
Fluorobenzene SCHEMBL27300498 0.84 NFE2L2 (0.46) ALDH1A1LMNANFE2L2
Formamide SCHEMBL28161914 0.79 CES2 (0.43) CES2CES1CA1CA2CA7
SCHEMBL27517155 0.79 CES2 (0.43) CES2CES1CA1CA9IDO1
Formic Acid SCHEMBL27369254 0.79 CES2 (0.50) CES2CES1CA1CA2CA7
SCHEMBL13499 0.76
SCHEMBL10306547 0.73
SCHEMBL2964 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 127 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106831814-B A kind of thieno [3,2-d] miazines HIV-1 reverse transcriptase inhibitor and its preparation method and application 山东大学 2018-11-23 CN claimed
CN-108484577-A A kind of pyrimidine-quinolones heterocomplex and its preparation method and application 复旦大学 2018-09-04 CN claimed
CN-107376875-A A kind of preparation and application of the beta cyclodextrin porous material with quick adsorption ability 湖南理工学院 2017-11-24 CN claimed
CN-106831814-A A kind of thieno [3,2 d] RTIs of miazines HIV 1 and its preparation method and application 山东大学 2017-06-13 CN claimed
CN-1785993-B Preparation and use of non-natural isocoumarin derivatives UNIV NANKAI 2012-03-14 CN claimed
CN-105683157-B Sulfonamides as sodium channel modulators 沃泰克斯药物股份有限公司 2019-07-19 CN disclosed
CN-104926733-B Compound as ROR gamma modulators 北京韩美药品有限公司 2019-05-10 CN disclosed
CN-105209458-B It is novel that there is the active 1,2,4- oxadiazole compound of resisting gram-positive pathogen 米兰比可卡大学 2019-01-04 CN disclosed
CN-109071457-A Inhibitors of indoleamine 2, 3-dioxygenase 荷兰转化研究中心有限责任公司 2018-12-21 CN disclosed
CN-108947868-A The preparation process of one kind 2,4- difluorobenzonilyile 山东师范大学 2018-12-07 CN disclosed
CN-106831814-B A kind of thieno [3,2-d] miazines HIV-1 reverse transcriptase inhibitor and its preparation method and application 山东大学 2018-11-23 CN disclosed
CN-108698982-A FLUORINE ATOM-CONTAINING COMPOUND AND USE THEREOF 日产化学工业株式会社 2018-10-23 CN disclosed
CN-1228695-A Substituted 1,2,3,4-tetrahydro-2-dibenzofuranamines and 2-aminocyclohepta [b] benzofurans LILLY CO ELI (US) 1999-09-15 CN disclosed
CN-1216986-A Isoxazole derivatives SANKYO CO (JP) 1999-05-19 CN disclosed
CN-1214039-A Carbamoyloxy derivatives of mutiline and their use as antibacterials SMITHKLINE BEECHAM PLC (GB) 1999-04-14 CN disclosed
CN-1160352-A Diaza * -oxindoles as phosphodiesterase IV inhibitors JOUVEINAL INST RECH (FR) 1997-09-24 CN disclosed
CN-1106802-A Tricyclic benzazepines (aza *) vasopressin antagonists AMERICAN CYANAMID CO (US) 1995-08-16 CN disclosed
CN-1023602-C Antipsychotic 3-piperazinylbenzazole derivs. JANSSEN PHARMACEUTICA NV (BE) 1994-01-26 CN disclosed
CN-1040194-A Psycholeptic 3-piperazinyl indole derivatives JANSSEN PHARMACEUTICA NV (BE) 1990-03-07 CN disclosed
CN-88103277-A Novel N-alkane sulfonyl aniline derivatives and preparation method thereof and the pharmaceutical composition that comprises this material 1988-12-07 CN disclosed