SCHEMBL2730786

SCHEMBL2730786

C=CC(=O)OCCn1c(=O)n(C)c(=O)n(CCOC(=O)C=C)c1=O

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.46
HPGD P15428 1/20 0.46
ALDH1A1 P00352 5/20 0.46
TP53 P04637 3/20 0.46
HIF1A Q16665 3/20 0.46
CYP3A4 P08684 3/20 0.46
HSD17B10 Q99714 1/20 0.46
THRB P10828 2/20 0.39
ADORA2B P29275 1/20 0.37
GAA P10253 2/20 0.35
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34
POLB P06746 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
PLA2G4A P47712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2730490 0.94 TSHR (0.49) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL42549 0.93 TSHR (0.52) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL2732955 0.90 TSHR (0.38) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL19117419 0.88 ALDH1A1 (0.50) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL14370783 0.88 TSHR (0.44) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL16545857 0.86 TSHR (0.49) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL25433797 0.86 TSHR (0.46) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL776295 0.86 TSHR (0.55) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL230828 0.86 TSHR (0.55) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL17589483 0.86 TSHR (0.50) TSHRHPGDALDH1A1TP53HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2635279-A2 CHEMICAL COMPOUNDS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2013-09-11 EP disclosed
EP-1698644-B1 FLUORINE-CONTAINING PHOTOCURING COMPOSITION DAINIPPON INK & CHEMICALS (JP) 2013-02-27 EP disclosed
WO-2012061557-A2 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2012-05-10 WO disclosed
JP-2011236175-A N-METHYL ISOCYANURATE COMPOUND SHIKOKU CHEM CORP 2011-11-24 JP disclosed
US-20070066779-A1 Fluorine-containing photocurable composition DIC CORPORATION (JP) 2007-03-22 US disclosed