SCHEMBL27309672

SCHEMBL27309672

CC(C)(C)OC(=O)Nc1ccc(Oc2ccnc(N3CCC(C(F)(F)F)C3)c2)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 9/20 0.44
KDR P35968 6/20 0.41
BRAF P15056 4/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
RORC P51449 1/20 0.40
ESRRA P11474 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30885063 1.00 MALT1 (0.44) MALT1KDRBRAFKDM4EMAPT
SCHEMBL27096932 0.89 MALT1 (0.45) MALT1KDRBRAFKDM4EMAPT
SCHEMBL30729915 0.87 NPC1 (0.46) MALT1KDRBRAFKDM4EMAPT
SCHEMBL27096974 0.79 MAP4K4 (0.41) MALT1KDM4EMAPTALDH1A1
SCHEMBL30729909 0.79 MAP4K4 (0.41) MALT1KDM4EMAPTALDH1A1
SCHEMBL30729912 0.78 ALDH1A1 (0.49) KDRBRAFMAPTRORCESRRA
SCHEMBL27305474 0.78 ALDH1A1 (0.49) KDRBRAFMAPTRORCESRRA
SCHEMBL30885060 0.75 KDR (0.57) KDRBRAF
SCHEMBL27305478 0.75 KDR (0.57) KDRBRAF
SCHEMBL29834832 0.72 MAP4K4 (0.39) KDRBRAFKDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024026056-A2 HETEROARYL COMPOUNDS AS EGFR INHIBITORS AND THEIR USES ACCUTAR BIOTECHNOLOGY, INC. (US) 2024-02-01 WO disclosed