SCHEMBL27316732

SCHEMBL27316732

CN1CCC(c2c[nH]c3ccc(CCC(=O)C=O)cc23)CC1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 14/20 0.62
HTR1B P28222 13/20 0.62
HTR1A P08908 4/20 0.62
HTR1F P30939 4/20 0.59
MAPT P10636 1/20 0.58
BLM P54132 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
THPO P40225 1/20 0.58
APP P05067 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27455068 0.94 HTR1D (0.55) HTR1DHTR1BHTR1AHTR1FMAPT
SCHEMBL9764535 0.87 HTR1D (0.64) HTR1DHTR1BHTR1AHTR1FMAPT
SCHEMBL8915046 0.86 HTR1D (0.63) HTR1DHTR1BHTR1AHTR1FMAPT
SCHEMBL27290426 0.86 NMT2 (0.55) HTR1DHTR1BHTR1AHTR1FAPP
SCHEMBL9764437 0.85 HTR1D (0.68) HTR1DHTR1BHTR1AHTR1FMAPT
Oxalic Acid SCHEMBL9764572 0.82 HTR1D (0.64) HTR1DHTR1BHTR1AHTR1FMAPT
SCHEMBL13234805 0.82 HTR1D (0.69) HTR1DHTR1BHTR1AHTR1FMAPT
SCHEMBL27294918 0.82 NMT2 (0.48) HTR1DHTR1BHTR1AHTR1FAPP
SCHEMBL9764751 0.80 HTR1D (0.65) HTR1DHTR1BHTR1AHTR1FMAPT
SCHEMBL27328413 0.80 HTR1D (0.47) HTR1DHTR1BHTR1AHTR1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1161967-A Preparation method for imidazole derivatives MERCK SHARP & DOHME (GB) 1997-10-15 CN claimed
CN-1128617-C Prepration method for medicinal composition containing triazolyl derivative MERCK SHARP & DOHME (GB) 2003-11-26 CN disclosed
CN-1061654-C Tetrazole derivatives and process for preparation thereof MERCK SHARP & DOHME (GB) 2001-02-07 CN disclosed
CN-1038681-C Triazole derivatives and their use as fungicides MERCK SHARP DOHME LTD (GB) 1998-06-10 CN disclosed
CN-1161967-A Preparation method for imidazole derivatives MERCK SHARP & DOHME (GB) 1997-10-15 CN disclosed
CN-1161834-A Prepration method for medicinal composition containing triazolyl derivative MERCK SHARP & DOHME (GB) 1997-10-15 CN disclosed
CN-1157821-A Process for preparation of tetrazole derivatives MERCK SHARP & DOHME (DE) 1997-08-27 CN disclosed