SCHEMBL27320400

SCHEMBL27320400

CCC(=O)c1cc(Br)c(OCCCBr)c(Br)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 6/20 0.48
THRA P10827 5/20 0.48
KLK1 P06870 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 2/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HRH3 Q9Y5N1 2/20 0.40
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
PPARA Q07869 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ESR1 P03372 1/20 0.39
NR1H4 Q96RI1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545057 0.83 KLK1 (0.47) THRBTHRAKLK1SMN1; SMN2ALDH1A1
SCHEMBL27323262 0.80 THRA (0.56) THRBTHRASMN1; SMN2ALDH1A1MEN1
SCHEMBL11027108 0.78 PPARG (0.40) THRBTHRASMN1; SMN2ALDH1A1MEN1
SCHEMBL26810030 0.78 TPMT (0.51) SMN1; SMN2ALDH1A1MEN1KMT2AKDM4E
SCHEMBL1334249 0.73 L3MBTL1 (0.58) THRBTHRASMN1; SMN2MEN1KMT2A
SCHEMBL7636855 0.73 KMT2A (0.49) THRBTHRAKLK1SMN1; SMN2ALDH1A1
SCHEMBL12370664 0.73 KLK1 (0.44) THRBTHRAKLK1ALDH1A1MEN1
SCHEMBL28031444 0.73 HRH3 (0.40) THRBTHRAKLK1SMN1; SMN2ALDH1A1
SCHEMBL8430188 0.72 TSHR (0.66) SMN1; SMN2ALDH1A1MEN1KMT2AKDM4E
SCHEMBL31063303 0.71 NCOA1 (0.46) SMN1; SMN2ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1086387-C N- (aryloxyalkyl) heteroarylpiperidines and heteroarylpiperazines, their preparation and their use as pharmaceuticals HOECHST MARION ROUSSEL INC (US) 2002-06-19 CN disclosed
CN-1048037-A N- (aryloxyalkyl) heteroarylpiperidines and heteroarylpiperazines, their preparation and their use as pharmaceuticals HOECHST ROUSSEL PHARMA (US) 1990-12-26 CN disclosed