SCHEMBL2732046

SCHEMBL2732046

Oc1ccc(-c2onc(-c3ccccc3Cl)c2-c2cccc(F)c2F)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
GPBAR1 Q8TDU6 2/20 0.39
DUSP3 P51452 3/20 0.39
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.37
ATM Q13315 1/20 0.37
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
HSD17B10 Q99714 1/20 0.36
USP7 Q93009 1/20 0.36
TSHR P16473 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MEN1 O00255 1/20 0.35
GFER P55789 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2732508 0.93 PTGS1 (0.45) PTGS1PTGS2GPBAR1DUSP3ALDH1A1
SCHEMBL2730709 0.88 PTGS1 (0.47) PTGS1PTGS2GPBAR1DUSP3ALDH1A1
SCHEMBL2730369 0.87 PTGS1 (0.41) PTGS1PTGS2GPBAR1DUSP3ALDH1A1
SCHEMBL2730611 0.87 LMNA (0.45) PTGS1PTGS2GPBAR1DUSP3ALDH1A1
SCHEMBL2730713 0.84 LMNA (0.45) PTGS1GPBAR1DUSP3ALDH1A1MAPT
SCHEMBL2729864 0.84 PTGS1 (0.41) PTGS1PTGS2GPBAR1DUSP3ALDH1A1
SCHEMBL2729879 0.84 PTGS1 (0.41) PTGS1PTGS2GPBAR1DUSP3ALDH1A1
SCHEMBL2730191 0.83 PTGS1 (0.43) PTGS1PTGS2GPBAR1DUSP3ALDH1A1
SCHEMBL2730299 0.83 PTGS1 (0.51) PTGS1PTGS2GPBAR1DUSP3ALDH1A1
SCHEMBL2732395 0.82 PTGS1 (0.59) PTGS1PTGS2DUSP3ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052395-A1 ISOXAZOLE DERIVATIVES USED AS OESTROGEN MODULATORS N. V. ORGANON (NL) 2012-04-26 WO disclosed
WO-2012052395-A1 ISOXAZOLE DERIVATIVES USED AS OESTROGEN MODULATORS N. V. ORGANON (NL) 2012-04-26 WO disclosed