SCHEMBL2732065

SCHEMBL2732065

CC[C@@H](N)c1ccccc1-c1c(C(=O)O)n(S(=O)(=O)c2ccccc2)c2ccc(OCc3ccccc3)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.42
HDAC1 Q13547 2/20 0.40
BCL2 P10415 1/20 0.40
BID P55957 1/20 0.40
MCL1 Q07820 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
EDNRB P24530 4/20 0.40
EDNRA P25101 4/20 0.40
ACLY P53396 1/20 0.39
SRD5A2 P31213 1/20 0.39
PSEN1 P49768 3/20 0.39
PSEN2 P49810 3/20 0.39
APH1B Q8WW43 3/20 0.39
NCSTN Q92542 3/20 0.39
APH1A Q96BI3 3/20 0.39
PSENEN Q9NZ42 3/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2733056 1.00 HTR6 (0.42) HTR6HDAC1BCL2BIDMCL1
SCHEMBL2733167 0.87 HTR6 (0.40) HTR6HDAC1BCL2BIDMCL1
SCHEMBL2732415 0.81 MEN1 (0.45) HTR6HDAC1BCL2BIDMCL1
SCHEMBL2724860 0.77 ACLY (0.39) HTR6ACLYPSEN1PSEN2APH1B
SCHEMBL2731882 0.77 HTR6 (0.48) HTR6HDAC1BCL2BIDMCL1
SCHEMBL2732312 0.75 HTR6 (0.39) HTR6HDAC1BCL2BIDMCL1
SCHEMBL2732313 0.75 HTR6 (0.39) HTR6HDAC1BCL2BIDMCL1
SCHEMBL10064904 0.73 PSEN1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2733172 0.70 ACLY (0.37) HTR6ACLYPSEN1PSEN2APH1B
SCHEMBL2726604 0.70 ACLY (0.41) HTR6ACLYPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059568-A1 NOVEL WATER-SOLUBLE INDOLOBENZAZEPINE MOLECULES DEMONSTRATING ANTIMITOTIC, ANTIVASCULAR, AND ANTITUMOR ACTIVITIES IN VIVO CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2012-05-10 WO disclosed