SCHEMBL27328403

SCHEMBL27328403

CC1CC(c2c[nH]c3ccc(-n4ccnn4)cc23)CN1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 6/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36
GABRE P78334 1/20 0.36
GABRA6 Q16445 1/20 0.36
GABRG1 Q8N1C3 1/20 0.36
GABRG3 Q99928 1/20 0.36
GABRQ Q9UN88 1/20 0.36
SLC6A4 P31645 7/20 0.35
HTR1B P28222 6/20 0.35
HTR1A P08908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27308222 0.80 HTR1D (0.42) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL8784287 0.80 HTR1D (0.58) HTR1BHTR1AHTR1DCYP1A2CYP3A4
SCHEMBL8783770 0.80 HTR2C (0.52) NOTUMGABRPGABRDGABRA1GABRB1
SCHEMBL27343954 0.80 HTR1A (0.50) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL8784524 0.78 KDM4E (0.58) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL8901002 0.77 CYP2D6 (0.43) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL31130003 0.73 NOTUM (0.50) NOTUMHTR1BHTR1AHTR1D
SCHEMBL27343955 0.73 HTR1A (0.53) SLC6A4HTR1BHTR1AHTR1D
SCHEMBL27327140 0.72 HTR1A (0.53) HTR1BHTR1AHTR1D
SCHEMBL27287897 0.67 HTR1D (0.53) SLC6A4HTR1BHTR1AHTR2AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1038681-C Triazole derivatives and their use as fungicides MERCK SHARP DOHME LTD (GB) 1998-06-10 CN claimed
CN-1061654-C Tetrazole derivatives and process for preparation thereof MERCK SHARP & DOHME (GB) 2001-02-07 CN disclosed
CN-1060479-C Preparation method for imidazole derivatives MERCK SHARP & DOHME (GB) 2001-01-10 CN disclosed
CN-1038681-C Triazole derivatives and their use as fungicides MERCK SHARP DOHME LTD (GB) 1998-06-10 CN disclosed
CN-1161967-A Preparation method for imidazole derivatives MERCK SHARP & DOHME (GB) 1997-10-15 CN disclosed
CN-1157821-A Process for preparation of tetrazole derivatives MERCK SHARP & DOHME (DE) 1997-08-27 CN disclosed