SCHEMBL8901002

SCHEMBL8901002

CCN1CCC(c2c[nH]c3ccc(-n4ccnn4)cc23)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.43
KDM4E B2RXH2 1/20 0.42
ATM Q13315 1/20 0.42
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
OPRM1 P35372 2/20 0.41
OPRK1 P41145 2/20 0.41
OPRL1 P41146 2/20 0.41
HTR1D P28221 2/20 0.41
HTR1B P28222 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
THPO P40225 1/20 0.41
GABRP O00591 2/20 0.41
GABRD O14764 2/20 0.41
GABRA1 P14867 2/20 0.41
GABRB1 P18505 2/20 0.41
GABRG2 P18507 2/20 0.41
GABRB3 P28472 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8784524 0.87 KDM4E (0.58) CYP2D6KDM4EATMNOS3NOS1
SCHEMBL8784287 0.85 HTR1D (0.58) CYP2D6KDM4EATMHTR1DHTR1B
SCHEMBL8783770 0.80 HTR2C (0.52) CYP2D6NOS3NOS1HTR1DHTR1B
SCHEMBL27328403 0.77 NOTUM (0.36) CYP2D6HTR1DHTR1BCYP1A2CYP3A4
SCHEMBL19210848 0.76 KDM4E (0.70) CYP2D6KDM4EATMSLC6A4
SCHEMBL8099607 0.73 PIM1 (0.45) CYP2D6KDM4EATMNOS3NOS1
SCHEMBL31130003 0.72 NOTUM (0.50) ATMHTR1DHTR1B
SCHEMBL7489311 0.70 HTR1D (0.74) CYP2D6NOS3NOS1OPRM1OPRK1
SCHEMBL25759842 0.69 ADRA1D (0.67) CYP2D6KDM4EATMSLC6A4
SCHEMBL8572226 0.69 KDM4E (0.60) CYP2D6KDM4EATMNOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602162-A TREATMENT AND/OR PREVENTION OF MIGRAINE MERCK, SHARP & DOHME LTD. (GB) 1997-02-11 US disclosed