SCHEMBL2733261

SCHEMBL2733261

O=C(O)c1c(I)c2ccccc2n1I

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
POLB P06746 3/20 0.40
THRB P10828 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
FABP3 P05413 2/20 0.39
FABP4 P15090 2/20 0.39
FABP5 Q01469 2/20 0.39
KDM4E B2RXH2 3/20 0.39
FOLH1 Q04609 3/20 0.39
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
LDHA P00338 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
ALOX12 P18054 1/20 0.38
ATIC P31939 1/20 0.38
NR4A1 P22736 1/20 0.37
NR4A2 P43354 1/20 0.37
NR4A3 Q92570 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689614 0.80 KDM4E (0.50) POLBL3MBTL1KDM4ETSHREGFR
SCHEMBL2724380 0.76 KDM4E (0.54) ALDH1A1POLBTHRBL3MBTL1KDM4E
SCHEMBL27967615 0.75 FOLH1 (0.62) ALDH1A1POLBKDM4EFOLH1HSD17B10
SCHEMBL2732076 0.74 FABP3 (0.50) FABP3FABP4FABP5LMNAMEN1
SCHEMBL27967763 0.72 PGR (0.52) ALDH1A1
SCHEMBL20115109 0.70 KDM4E (0.52) ALDH1A1POLBL3MBTL1FABP3FABP4
SCHEMBL7111400 0.70 EDNRA (0.56) ALDH1A1KDM4EFOLH1HPGDLMNA
SCHEMBL16009974 0.69 POLB (0.48) ALDH1A1POLBKDM4EHPGDHSD17B10
SCHEMBL13357151 0.67 GPR3 (0.52) ALDH1A1POLBL3MBTL1FABP3FABP4
SCHEMBL21311770 0.65 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059568-A1 NOVEL WATER-SOLUBLE INDOLOBENZAZEPINE MOLECULES DEMONSTRATING ANTIMITOTIC, ANTIVASCULAR, AND ANTITUMOR ACTIVITIES IN VIVO CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2012-05-10 WO disclosed