SCHEMBL2733263

SCHEMBL2733263

O=C(O)c1[nH]c2cccc(I)c2c1I

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 3/20 0.61
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.38
PARP1 P09874 1/20 0.38
FOLH1 Q04609 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2724384 0.80 GPR17 (0.49) GPR17KDM4EALDH1A1HPGDMEN1
SCHEMBL9452228 0.75 HPGD (0.57) GPR17KDM4EALDH1A1HPGDMEN1
SCHEMBL2724876 0.74 KDM4E (0.61) KDM4EALDH1A1HPGDMEN1POLB
SCHEMBL31245675 0.74 KDM4E (0.61) KDM4EALDH1A1HPGDMEN1POLB
SCHEMBL5027261 0.73 KDM4E (0.47) GPR17KDM4EALDH1A1PARP1
SCHEMBL48966 0.69 IMPDH2 (0.47) GPR17KDM4EALDH1A1HPGDMEN1
SCHEMBL27760409 0.69 PARP1 (0.54) GPR17KDM4EALDH1A1HPGDPARP1
SCHEMBL29350550 0.69 IMPDH2 (0.47) GPR17KDM4EALDH1A1HPGDMEN1
SCHEMBL8752557 0.69 GPR17 (0.58) GPR17HPGDMEN1KMT2A
SCHEMBL15516976 0.68 MCL1 (0.44) GPR17KDM4EALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059568-A1 NOVEL WATER-SOLUBLE INDOLOBENZAZEPINE MOLECULES DEMONSTRATING ANTIMITOTIC, ANTIVASCULAR, AND ANTITUMOR ACTIVITIES IN VIVO CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2012-05-10 WO disclosed