SCHEMBL2733602

SCHEMBL2733602

CCN(CC)C(=O)c1ccc(Br)cc1S(C)(=O)=O

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.49
HSP90AA1 P07900 3/20 0.42
HSP90AB1 P08238 3/20 0.42
ALDH1A1 P00352 3/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.41
LMNA P02545 2/20 0.41
TSHR P16473 1/20 0.41
HPGD P15428 2/20 0.41
KEAP1 Q14145 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GFER P55789 1/20 0.38
TSPO P30536 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1369724 0.84 PTGDR2 (0.48) USP2HSP90AA1HSP90AB1ALDH1A1RAB9A
SCHEMBL471624 0.78 USP2 (0.54) USP2HSP90AA1HSP90AB1ALDH1A1RAB9A
SCHEMBL2170651 0.78 HPGD (0.57) USP2HSP90AA1HSP90AB1ALDH1A1RAB9A
SCHEMBL1369782 0.77 PTGDR2 (0.43) USP2HSP90AA1HSP90AB1ALDH1A1RAB9A
SCHEMBL1085171 0.77 KDM4E (0.47) ALDH1A1MAPK1LMNA
SCHEMBL3552169 0.76 USP2 (0.52) USP2HSP90AA1HSP90AB1ALDH1A1RAB9A
SCHEMBL3341268 0.76 DGAT1 (0.54) USP2HSP90AA1HSP90AB1ALDH1A1RAB9A
SCHEMBL3472808 0.76 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2MAPK1L3MBTL1LMNA
SCHEMBL9173722 0.76 WDR5 (0.42) ALDH1A1HPGD
SCHEMBL17505003 0.76 DGAT1 (0.53) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632464-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2013-09-04 EP disclosed
WO-2012058134-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed