SCHEMBL27346293

SCHEMBL27346293

Nc1cccc(-c2ncccn2)c1S(N)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.40
CA2 P00918 6/20 0.40
CA9 Q16790 4/20 0.40
CA12 O43570 3/20 0.40
MAPK1 P28482 1/20 0.39
CYP2C9 P11712 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
PTPRC P08575 1/20 0.35
ADORA2A P29274 1/20 0.35
KMT2A Q03164 2/20 0.35
KDM1A O60341 1/20 0.35
TDP2 O95551 2/20 0.34
NSD2 O96028 2/20 0.34
PAX8 Q06710 2/20 0.34
ABL1 P00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27281513 0.81 TDO2 (0.41) CA1CA2CA9CA12MAPK1
SCHEMBL8697134 0.79 CA1 (0.42) CA1CA2CA9CA12MAPK1
SCHEMBL22502056 0.77 NAPRT (0.45) CA1CA2CA9BLMTDP1
SCHEMBL28026576 0.76 CA2 (0.54) CA1CA2CA9CA12CYP2C9
SCHEMBL27685705 0.76 ADORA2A (0.44) CA1CA2CA9CA12CYP2C9
SCHEMBL6564249 0.74 ALDH1A1 (0.54) CA1CA2CA9CA12MAPK1
SCHEMBL1232419 0.72 ALDH1A1 (0.57) ADORA2AKMT2AMEN1TDP1GAA
SCHEMBL1094361 0.72 CA1 (0.50) CA1CA2CA9CA12MAPK1
SCHEMBL1319393 0.71 ALDH1A1 (0.56) CYP2C9KMT2ATDP2MEN1BLM
SCHEMBL11882081 0.70 CA2 (0.50) CA1CA2CA9CA12CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107250135-A The preparation method of long-acting dipeptidy peptidase in inhibitors, purposes and its intermediate 四川科伦药物研究院有限公司 2017-10-13 CN disclosed
CN-1407973-A Butynediol Derivatives ACTELION PHARMACEUTICALS LTD (CH) 2003-04-02 CN disclosed
CN-1052484-C 5-Alkoxy [1,2,4] triazolo [1,5,-C] pyrimidine -2[3H]-thione compounds and their use DOW AGROSCIENCES LLC (US) 2000-05-17 CN disclosed
CN-1243514-A Sulfonamide derivatives KOREA RES INST CHEM TECH (KR) 2000-02-02 CN disclosed
CN-1205336-A 5-Alkoxy [1,2,4] triazolo [1,5,-C] pyrimidine -2[3H]-thione compounds and their use DOW AGROSCIENCES LLC (US) 1999-01-20 CN disclosed
CN-1041092-C 5-alkoxy [1, 2, 4] triazolo [1, 5-C ] pyrimidine-2 (3H) -thiones and their use DOEWLANCO SCIENCE CO (US) 1998-12-09 CN disclosed
CN-1033806-C Herbicidal composition DOWELANCO (US) 1997-01-15 CN disclosed
CN-1134223-A Method for controling needless plant DOWELANCO (US) 1996-10-30 CN disclosed
CN-1115983-A 5-alkoxy [1, 2, 4] triazolo [1, 5-C ] pyrimidine-2 (3H) -thiones and their use DOWELANCO (US) 1996-01-31 CN disclosed
CN-1068824-A N-pyrazolyl-1, 2, 4-triazolo [1, 5-c ] pyrimidine-2-sulfonamides as herbicides DOWELANCO (US) 1993-02-10 CN disclosed