SCHEMBL27355398

SCHEMBL27355398

CCOC(=O)c1nc(Cc2ccc3c(c2)OCO3)c2c(N)c(Cl)ccc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
HSD17B10 Q99714 5/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
LMNA P02545 3/20 0.43
ALOX15 P16050 2/20 0.43
MAPT P10636 2/20 0.43
USP2 O75604 1/20 0.43
PDE5A O76074 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
SIRT3 Q9NTG7 1/20 0.41
CHRM4 P08173 2/20 0.41
LTB4R Q15722 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
KDM4E B2RXH2 2/20 0.40
TP53 P04637 2/20 0.40
HPGD P15428 4/20 0.40
MAPK1 P28482 2/20 0.40
PRKCI P41743 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27382274 0.84 CHRM4 (0.39) ALDH1A1HSD17B10MEN1KMT2ALMNA
SCHEMBL27452402 0.83 CHRM4 (0.38) ALDH1A1HSD17B10MEN1KMT2ALMNA
SCHEMBL27364630 0.83 CHRM4 (0.38) ALDH1A1HSD17B10MEN1KMT2ALMNA
SCHEMBL27531812 0.82 MEN1 (0.42) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL27377273 0.81 ALDH1A1 (0.42) ALDH1A1HSD17B10MEN1KMT2ALMNA
SCHEMBL7794556 0.81 ALDH1A1 (0.46) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL8862704 0.80 LTB4R (0.46) ALDH1A1HSD17B10CHRM4LTB4R
SCHEMBL27379780 0.80 SLC2A1 (0.47) ALDH1A1HSD17B10LTB4R
SCHEMBL9094776 0.79 LTB4R (0.41) ALDH1A1HSD17B10LMNACHRM4LTB4R
SCHEMBL7794741 0.79 CHRM4 (0.42) ALDH1A1HSD17B10MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1071164-A Nitrogen-containing heterocycle compound EISAI CO LTD (JP) 1993-04-21 CN disclosed