SCHEMBL27360404

SCHEMBL27360404

Nc1c(Cl)cc(C(=O)ON2CCCCC2)c2c1CCO2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 5/20 0.50
HTR3A P46098 4/20 0.50
HTR3E A5X5Y0 2/20 0.50
HTR3B O95264 2/20 0.50
HTR3D Q70Z44 2/20 0.50
HTR3C Q8WXA8 2/20 0.50
ADRA2C P18825 2/20 0.47
ADRA1A P35348 2/20 0.47
HTR1A P08908 1/20 0.47
ACHE P22303 1/20 0.47
PTGS1 P23219 1/20 0.47
KCNH2 Q12809 1/20 0.47
HTR2C P28335 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
LMNA P02545 1/20 0.40
ADRA2A P08913 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alcohol SCHEMBL8799335 0.94 HTR4 (0.48) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL7355300 0.81 HTR4 (0.55) HTR4HTR3AHTR3EHTR3BHTR3D
Hydrochloric Acid SCHEMBL7361117 0.80 HTR4 (0.54) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL5042523 0.80 HTR4 (0.54) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL7365594 0.79 HTR4 (0.60) HTR4HTR3AHTR3EHTR3BHTR3D
Hydrochloric Acid SCHEMBL7363349 0.79 HTR4 (0.59) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL27384092 0.78 HTR4 (0.38) HTR4HTR3AHTR3EHTR3BHTR3D
Hydrochloric Acid SCHEMBL7361288 0.78 HTR4 (0.47) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL8509459 0.78 HTR4 (0.52) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL1502018 0.76 HTR4 (0.51) HTR4HTR3AHTR3EHTR3BHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1068881-C Phenyl-oxo-alkyl-(4-piperidinyl) benzoate derivs. JANSSEN PHARMACEUTICA NV (BE) 2001-07-25 CN disclosed
CN-1068880-C N-substituted piperidinyl bicyclic benzoate derivatives JANSSEN PHARMACEUTICA NV (BE) 2001-07-25 CN disclosed
CN-1166171-A N-substituted piperidinyl bicyclic benzoate derivatives JANSSEN PHARMACEUTICA NV (BE) 1997-11-26 CN disclosed
CN-1160401-A Phenyl-oxo-alkyl- (4-piperidinyl) benzoate derivatives JANSSEN PHARMACEUTICA NV (BE) 1997-09-24 CN disclosed