SCHEMBL27362345

SCHEMBL27362345

Cn1cc(-c2ccccc2)c2c[c]ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.49
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
IMPDH2 P12268 2/20 0.43
GSK3B P49841 2/20 0.40
ASH1L Q9NR48 1/20 0.40
SCN9A Q15858 1/20 0.39
NFATC1 O95644 1/20 0.38
DYRK1A Q13627 1/20 0.38
CCNE2 O96020 1/20 0.37
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CCNE1 P24864 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695819 0.87 BRD4 (0.49) BRD4KDM4ENPC1ALDH1A1CYP1A2
SCHEMBL3131200 0.79 IMPDH2 (0.57) BRD4KDM4ENPC1ALDH1A1CYP1A2
SCHEMBL733151 0.79 DYRK1A (0.47) BRD4KDM4EHPGDGSK3BDYRK1A
SCHEMBL3149953 0.79 IMPDH2 (0.53) BRD4KDM4ENPC1ALDH1A1CYP1A2
SCHEMBL1310255 0.78 IMPDH2 (0.64) BRD4KDM4ENPC1ALDH1A1CYP1A2
SCHEMBL2596719 0.73 IMPDH2 (0.35) ALDH1A1IMPDH2GPR84
SCHEMBL25328590 0.72 IMPDH2 (0.34) ALDH1A1IMPDH2GSK3BGPR84NPSR1
SCHEMBL27736804 0.72 IMPDH2 (0.34) ALDH1A1IMPDH2CCNT1CDK9GPR84
SCHEMBL3482821 0.71 GPR84 (0.44) KDM4EALDH1A1HPGDIMPDH2GPR84
SCHEMBL695859 0.71 IDO1 (0.44) BRD4KDM4EALDH1A1IMPDH2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1073443-A Preparation method with macrolide of immunosuppressive activity MERCK & CO INC (US) 1993-06-23 CN disclosed