SCHEMBL27362971

SCHEMBL27362971

CCOC(=O)c1cn2cc(-c3ccc(NS(C)(=O)=O)cc3)nc2s1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.51
RECQL P46063 1/20 0.51
TP53 P04637 5/20 0.47
RXFP1 Q9HBX9 3/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 4/20 0.44
MMP2 P08253 1/20 0.43
MMP13 P45452 1/20 0.43
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
ACR P10323 1/20 0.40
MTOR P42345 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27361295 0.84 KMT2A (0.51) HPGDTP53RXFP1MEN1KMT2A
SCHEMBL29924707 0.84 MAPT (0.53) HPGDTP53MEN1KMT2AMAPT
SCHEMBL27362964 0.82 MAPT (0.39) HPGDTP53RXFP1MEN1KMT2A
SCHEMBL22117098 0.82 SMN1; SMN2 (0.53) HPGDTP53MEN1KMT2AMAPT
SCHEMBL5017019 0.82 SMN1; SMN2 (0.51) HPGDTP53MEN1KMT2AMAPT
SCHEMBL27362958 0.80 MAPT (0.56) HPGDRECQLTP53RXFP1MEN1
SCHEMBL27362937 0.80 MAPT (0.59) HPGDRECQLTP53RXFP1MEN1
SCHEMBL29925367 0.74 SMN1; SMN2 (0.48) HPGDTP53MEN1KMT2AMAPT
SCHEMBL21760981 0.73 ALDH1A1 (0.43) HPGDMEN1KMT2AMAPTNPC1
SCHEMBL3059986 0.73 MAPT (0.48) HPGDTP53MAPTNPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023235753-A2 ALDH2 INHIBITORS AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-12-07 WO disclosed