SCHEMBL27362937

SCHEMBL27362937

CCOC(=O)c1csc2nc(-c3ccc(NS(C)(=O)=O)cc3)cn12

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.59
TP53 P04637 5/20 0.59
RXFP1 Q9HBX9 2/20 0.59
HPGD P15428 2/20 0.50
RECQL P46063 1/20 0.50
POLB P06746 2/20 0.46
PTGS2 P35354 1/20 0.44
FLT3 P36888 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
MMP2 P08253 1/20 0.42
MMP13 P45452 1/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27362934 0.85 MAPT (0.59) MAPTTP53RXFP1HPGDPOLB
SCHEMBL27362958 0.81 MAPT (0.56) MAPTTP53RXFP1HPGDRECQL
SCHEMBL27362971 0.80 HPGD (0.51) MAPTTP53RXFP1HPGDRECQL
SCHEMBL20538978 0.76 CDC7 (0.50) MAPTTP53HPGDPOLBPTGS2
SCHEMBL2624439 0.73 IDO1 (0.41) MAPTTP53RXFP1HPGDPTGS2
SCHEMBL2564662 0.72 IDO1 (0.43) MAPTTP53RXFP1PTGS2MEN1
SCHEMBL13470766 0.72 ALDH1A1 (0.43) MAPTTP53HPGDPOLBPTGS2
SCHEMBL11327747 0.71 GAA (0.45) MAPTHPGDPOLBMEN1KMT2A
SCHEMBL27361298 0.70 RAB9A (0.57) MAPTTP53RXFP1HPGDPOLB
SCHEMBL13470789 0.70 ALDH1A1 (0.40) MAPTTP53HPGDPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023235753-A2 ALDH2 INHIBITORS AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-12-07 WO disclosed