SCHEMBL27363963

SCHEMBL27363963

COC(=O)c1ccc(C#CC2(O)CCCC[C@@H]2OC)cc1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.43
MMP13 P45452 5/20 0.41
GRM5 P41594 5/20 0.40
MMP2 P08253 1/20 0.40
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
EPHX2 P34913 1/20 0.39
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27216857 1.00 PTPN11 (0.43) PTPN11MMP13GRM5MMP2NPC1
SCHEMBL27363438 0.96 PTPN11 (0.44) PTPN11MMP13GRM5MMP2NPC1
SCHEMBL30809918 0.89 MMP13 (0.48) MMP13GRM5MMP2ALDH1A1
SCHEMBL30809908 0.85 MMP13 (0.45) PTPN11MMP13GRM5MMP2ALDH1A1
SCHEMBL27364406 0.84 GRM5 (0.40) PTPN11GRM5ALDH1A1
SCHEMBL27363769 0.79 ALDH1A1 (0.55) PTPN11GRM5NPC1ALDH1A1SMN1; SMN2
SCHEMBL27363966 0.78 ALDH1A1 (0.57) PTPN11GRM5NPC1ALDH1A1SMN1; SMN2
SCHEMBL28516359 0.76 ALDH1A1 (0.52) PTPN11GRM5ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL4815450 0.73 PTPN11 (0.45) PTPN11NPC1ALDH1A1CYP2C19
SCHEMBL27365315 0.72 FFAR1 (0.51) PTPN11NPC1ALDH1A1SMN1; SMN2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024054624-A1 MODULATORS OF ALPHA-1 ANTITRYPSIN VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-03-14 WO disclosed