SCHEMBL27365091

SCHEMBL27365091

Cc1cccc(C2CCN(CC3CN(C)C3)CC2)c1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.54
DRD4 P21917 5/20 0.54
DRD3 P35462 4/20 0.54
DRD1 P21728 2/20 0.54
DRD5 P21918 2/20 0.54
CCR5 P51681 1/20 0.53
HTR2C P28335 2/20 0.48
HTR1A P08908 1/20 0.44
TRPV6 Q9H1D0 1/20 0.44
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27365089 0.89 DRD2 (0.51) DRD2DRD4DRD3DRD1DRD5
SCHEMBL27367007 0.85 DRD3 (0.56) DRD2DRD4DRD3DRD1DRD5
SCHEMBL27364866 0.82 DRD2 (0.46) DRD2DRD4DRD3CCR5
SCHEMBL15829965 0.81 DRD2 (0.60) DRD2DRD4DRD3DRD1DRD5
SCHEMBL11619057 0.80 HTR2C (0.61) DRD2DRD4DRD3DRD1DRD5
SCHEMBL27364231 0.78 DRD2 (0.52) DRD2DRD4DRD3DRD1DRD5
SCHEMBL12320891 0.78 SLC18A3 (0.67) DRD2DRD4DRD3DRD1DRD5
SCHEMBL30878617 0.78 DRD3 (0.65) DRD2DRD4DRD3DRD1DRD5
SCHEMBL27321176 0.77 HTR2C (0.55) DRD2DRD4DRD3DRD1DRD5
SCHEMBL7653412 0.76 DRD2 (0.52) DRD2DRD4DRD3DRD1DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024054591-A1 RAPIDLY ACCELERATED FIBROSARCOMA (RAF) DEGRADING COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. (US) 2024-03-14 WO disclosed