SCHEMBL27367381

SCHEMBL27367381

Cc1ccc(N2CC(CN3CCN(C4CC[N+](C)(C)CC4)CC3)C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
MEN1 O00255 4/20 0.37
L3MBTL3 Q96JM7 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27364619 0.85 KMT2A (0.42) KMT2AMEN1L3MBTL3L3MBTL1MAPT
SCHEMBL27368371 0.84 ADRB1 (0.45) KMT2AMEN1
SCHEMBL27366536 0.82 PDE10A (0.43) KMT2AMEN1MAPT
SCHEMBL27365606 0.77 MAPT (0.44) KMT2AMEN1MAPTNPSR1
SCHEMBL27367216 0.74 EBP (0.43)
SCHEMBL12082219 0.72 MAPT (0.51) KMT2AMEN1MAPTNPSR1
SCHEMBL20372819 0.71 MAPT (0.51) MAPTNPSR1
SCHEMBL27365359 0.70 ADRB1 (0.38) KMT2AMEN1MAPTNPSR1
SCHEMBL14924468 0.70 KMT2A (0.67) KMT2AL3MBTL3L3MBTL1MAPT
SCHEMBL81591 0.70 L3MBTL3 (0.57) KMT2AMEN1L3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024054591-A1 RAPIDLY ACCELERATED FIBROSARCOMA (RAF) DEGRADING COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. (US) 2024-03-14 WO disclosed