SCHEMBL27368090

SCHEMBL27368090

CC(=O)Oc1cc(CCBr)ccc1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.49
CFD P00746 2/20 0.44
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
ADORA3 P0DMS8 2/20 0.43
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
CCR5 P51681 1/20 0.43
PTGS2 P35354 4/20 0.42
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
GLA P06280 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ESR1 P03372 1/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
HMGB1 P09429 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27489237 0.89 BACE1 (0.51) BACE1CFDCYP4F2CYP4A11ADORA3
SCHEMBL11835902 0.83 BACE1 (0.44) BACE1CFDCYP4F2CYP4A11ADORA3
SCHEMBL28035132 0.83 BACE1 (0.51) BACE1CFDCYP4F2CYP4A11ADORA3
SCHEMBL27556516 0.81 HTR7 (0.44) CYP4F2CYP4A11KDM4EKMT2AALDH1A1
SCHEMBL7658162 0.81 CFD (0.53) CFDCYP4F2CYP4A11CCR5KDM4E
SCHEMBL27623501 0.78 CFD (0.59) CFDCYP4F2CYP4A11CCR5PTGS2
SCHEMBL10448896 0.77 BACE1 (0.41) BACE1CYP4F2CYP4A11ADORA3ADORA2A
SCHEMBL31273249 0.76 BACE1 (0.61) BACE1ADORA3ADORA2AADORA1KDM4E
SCHEMBL28022867 0.76 BACE1 (0.56) BACE1ADORA3ADORA2AADORA1PTGS2
SCHEMBL11835597 0.76 BACE1 (0.44) BACE1CFDCYP4F2CYP4A11ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1066070-A Promote the new benzo-fused lactams that tethelin discharges MERCK & CO INC (US) 1992-11-11 CN disclosed