SCHEMBL2737050

SCHEMBL2737050

CCOC(=O)c1ccc(-n2cc(N)c3cc(-c4ccc(O)c(Cl)c4)ccc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.46
CA12 O43570 3/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
CA7 P43166 2/20 0.41
CA14 Q9ULX7 2/20 0.41
SRC P12931 2/20 0.41
LCK P06239 1/20 0.41
KIT P10721 1/20 0.41
GABRA2 P47869 2/20 0.40
GABRB2 P47870 2/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAOA P21397 1/20 0.40
EGFR P00533 1/20 0.39
KDR P35968 1/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10207671 0.85 EGFR (0.48) SRCGABRA2GABRB2LMNAEGFR
SCHEMBL12309511 0.85
SCHEMBL2737105 0.83 CA12 (0.51) CA12CA1CA2CA9CA7
SCHEMBL2737123 0.80 HPGD (0.57) CHRNA7CA1CA2SRCLCK
SCHEMBL13594234 0.79 HDAC1 (0.48) SRCEGFRKDRALDH1A1TSHR
SCHEMBL2736511 0.79 HPGD (0.47) CA12CA1CA2CA9CA7
SCHEMBL2736546 0.78 LMNA (0.44) CHRNA7CA12CA1CA2CA9
SCHEMBL2737111 0.76 MAPT (0.49) SRCLMNAEGFRKDRHPGD
SCHEMBL2737112 0.75 TDP1 (0.47) GABRA2LMNAHPGDSMN1; SMN2TDP1
SCHEMBL2736681 0.74 SMN1; SMN2 (0.46) LMNACYP1A2CYP3A4MAOAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402314-A1 (Aza)indole derivative and use thereof for medical purposes Kissei Pharmaceutical Co., Ltd. (JP) 2012-01-04 EP disclosed