SCHEMBL27415403

SCHEMBL27415403

O=C1CC(c2ccc(Br)cc2)C(C(=O)O)N1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
LMNA P02545 2/20 0.46
NPSR1 Q6W5P4 1/20 0.44
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
FPR1 P21462 1/20 0.39
GPBAR1 Q8TDU6 1/20 0.38
KDM1A O60341 5/20 0.38
KCNH2 Q12809 2/20 0.38
MAOB P27338 2/20 0.38
RCOR1 Q9UKL0 2/20 0.38
KDM1B Q8NB78 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PLA2G1B P04054 1/20 0.35
GAPDH P04406 1/20 0.35
POLB P06746 1/20 0.35
HSPA1A P0DMV8 1/20 0.35
MIF P14174 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27415402 1.00 ALDH1A1 (0.46) ALDH1A1LMNANPSR1CYP2C9CYP2C19
SCHEMBL9745628 0.85 ALDH1A1 (0.59) ALDH1A1LMNANPSR1SMN1; SMN2
SCHEMBL9745446 0.85 ALDH1A1 (0.59) ALDH1A1LMNANPSR1SMN1; SMN2
SCHEMBL9745453 0.85 ALDH1A1 (0.59) ALDH1A1LMNANPSR1SMN1; SMN2
SCHEMBL27492314 0.84 ALDH1A1 (0.52) ALDH1A1LMNANPSR1KDM1AKCNH2
SCHEMBL16055833 0.84 ALDH1A1 (0.46) ALDH1A1LMNANPSR1FPR1GPBAR1
SCHEMBL27492313 0.84 ALDH1A1 (0.52) ALDH1A1LMNANPSR1KDM1AKCNH2
SCHEMBL27565973 0.79 ALDH1A1 (0.45) ALDH1A1LMNANPSR1SMN1; SMN2MEN1
SCHEMBL27565971 0.79 ALDH1A1 (0.45) ALDH1A1LMNANPSR1SMN1; SMN2MEN1
SCHEMBL18586607 0.76 LMNA (0.50) ALDH1A1LMNACYP2C9CYP2C19FPR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1210256-C Diacylhydrazine derivs. MERCK PATENT GMBH (DE) 2005-07-13 CN disclosed
CN-1117077-C 6-phenylpyridyl-2-amine derivatives useful as NOS inhibitors PFIZER (US) 2003-08-06 CN disclosed
CN-1360568-A Diacylhydrazine derivs. MERCK PATENT GMBH (DE) 2002-07-24 CN disclosed
CN-1239952-A 6-phenylpyridyl-2-amine derivatives useful as NOS inhibitors PFIZER (US) 1999-12-29 CN disclosed